SCHEMBL6984810

SCHEMBL6984810

CN(C(=O)c1ccc(Cl)cc1)c1cccc2c1N(C(=O)CCc1ccc(C#N)cc1)CCC2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 1/20 0.38
POLB P06746 1/20 0.38
DRD2 P14416 2/20 0.37
DRD4 P21917 2/20 0.37
CCR1 P32246 1/20 0.37
MCHR1 Q99705 1/20 0.36
AVPR2 P30518 2/20 0.36
AVPR1A P37288 2/20 0.36
IDO1 P14902 2/20 0.36
KCNH2 Q12809 2/20 0.36
CNR1 P21554 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
FPR1 P21462 2/20 0.34
FPR2 P25090 2/20 0.34
ITK Q08881 1/20 0.34
NSD2 O96028 1/20 0.34
OXTR P30559 1/20 0.34
RXRA P19793 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981987 0.92 PTGER4 (0.38) PTGER4AVPR2AVPR1AFPR1FPR2
SCHEMBL7409214 0.85 PTGER4 (0.38) PTGER4POLBDRD2DRD4CCR1
SCHEMBL6984734 0.84 AVPR2 (0.36) PTGER4AVPR2AVPR1AFPR1FPR2
SCHEMBL7958965 0.82 IDO1 (0.45) POLBDRD2DRD4AVPR2IDO1
SCHEMBL6986002 0.81 RXRA (0.45) PTGER4RXRARXRBRXRG
SCHEMBL7958782 0.80 IDO1 (0.45) POLBDRD2DRD4AVPR2IDO1
SCHEMBL6979942 0.80 TSHR (0.38) PTGER4AVPR2AVPR1AFPR1FPR2
SCHEMBL6986115 0.80 ITGB3 (0.40) PTGER4AVPR2AVPR1AOXTRRXRA
SCHEMBL6977636 0.79 ALDH1A1 (0.42)
SCHEMBL6986008 0.78 MEN1 (0.39) PTGER4AVPR2AVPR1AFPR1FPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed