SCHEMBL6977636

SCHEMBL6977636

CN(c1cccc2c1N(C(=O)CCc1ccc(C#N)cc1)CCC2)S(=O)(=O)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
NR3C1 P04150 2/20 0.40
TAS2R14 Q9NYV8 1/20 0.39
MEN1 O00255 2/20 0.39
HPGD P15428 2/20 0.39
KMT2A Q03164 2/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 2/20 0.39
MAPK1 P28482 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TSHR P16473 2/20 0.38
USP2 O75604 1/20 0.38
HSD17B10 Q99714 1/20 0.38
AR P10275 1/20 0.38
C5AR1 P21730 1/20 0.37
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6982667 0.90 NR3C1 (0.41) ALDH1A1NR3C1TAS2R14MEN1HPGD
SCHEMBL6981554 0.89 ALDH1A1 (0.44) ALDH1A1MEN1HPGDKMT2ALMNA
SCHEMBL6986002 0.88 RXRA (0.45) ALDH1A1TAS2R14MEN1HPGDKMT2A
SCHEMBL6987767 0.86 TP53 (0.42) ALDH1A1NR3C1LMNAGAAUSP2
SCHEMBL6982999 0.85 ALDH1A1 (0.41) ALDH1A1HPGDLMNAGAAMAPT
SCHEMBL6977634 0.85 NR3C1 (0.53) ALDH1A1NR3C1MEN1HPGDKMT2A
SCHEMBL6987632 0.85 ALDH1A1 (0.39) ALDH1A1NR3C1TAS2R14MEN1HPGD
SCHEMBL6981987 0.85 PTGER4 (0.38) ALDH1A1NR3C1MEN1HPGDKMT2A
SCHEMBL6983751 0.84 NR3C1 (0.40) ALDH1A1NR3C1MEN1HPGDKMT2A
SCHEMBL6986008 0.83 MEN1 (0.39) ALDH1A1MEN1HPGDKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed