SCHEMBL6984884

SCHEMBL6984884

Cc1c(C)c2c(c(C)c1N)CC(C)(CN1CCN(C(=O)c3ccc(Cl)cc3)CC1)O2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45
POLB P06746 1/20 0.42
KCNA5 P22460 2/20 0.41
LSS P48449 2/20 0.41
GPR183 P32249 1/20 0.41
LMNA P02545 1/20 0.40
DRD2 P14416 2/20 0.39
LDHA P00338 1/20 0.39
DRD3 P35462 1/20 0.39
PHGDH O43175 1/20 0.39
THRB P10828 1/20 0.39
KMT2A Q03164 2/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6984699 0.92 ALDH1A1 (0.40) KDM4EALDH1A1POLBKCNA5LMNA
SCHEMBL8579633 0.89 DRD3 (0.40) ALDH1A1LSSLMNADRD2DRD3
SCHEMBL6983343 0.89 DRD2 (0.46) ALDH1A1POLBKCNA5LSSDRD2
SCHEMBL6976774 0.88 CA12 (0.44) KDM4EALDH1A1POLBLMNAKMT2A
SCHEMBL6982084 0.84 ALDH1A1 (0.48) KDM4EALDH1A1MAPTPOLBLMNA
Hydrochloric Acid SCHEMBL6981668 0.83 SIGMAR1 (0.38) KDM4EALDH1A1MAPTPOLBLSS
SCHEMBL6978716 0.82 MEN1 (0.48) KDM4EALDH1A1LMNADRD2DRD3
SCHEMBL7097588 0.80 TP53 (0.36) KDM4EMAPTPOLBLMNADRD2
SCHEMBL6980270 0.80 CCR3 (0.42) DRD2DRD3
SCHEMBL6981792 0.79 POLB (0.47) KDM4EALDH1A1POLBLMNADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed