SCHEMBL6982084

SCHEMBL6982084

COc1ccc(C(=O)N2CCN(CC3(C)Cc4c(C)c(N)c(C)c(C)c4O3)CC2)cc1OC

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
POLB P06746 1/20 0.48
CYP2C19 P33261 1/20 0.48
KDM4E B2RXH2 4/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
KMT2A Q03164 2/20 0.46
GAA P10253 3/20 0.45
MAPT P10636 2/20 0.45
TSHR P16473 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
ATM Q13315 1/20 0.44
LMNA P02545 3/20 0.44
MEN1 O00255 1/20 0.44
TP53 P04637 2/20 0.43
HTT P42858 1/20 0.43
HPGD P15428 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983343 0.88 DRD2 (0.46) ALDH1A1POLBTSHRHPGD
SCHEMBL6978716 0.87 MEN1 (0.48) ALDH1A1KDM4ESMN1; SMN2KMT2ALMNA
SCHEMBL6984699 0.86 ALDH1A1 (0.40) ALDH1A1POLBKDM4ESMN1; SMN2KMT2A
SCHEMBL6981792 0.85 POLB (0.47) ALDH1A1POLBCYP2C19KDM4ESMN1; SMN2
SCHEMBL8579633 0.83 DRD3 (0.40) ALDH1A1SMN1; SMN2KMT2AGAALMNA
SCHEMBL6976774 0.82 CA12 (0.44) ALDH1A1POLBKDM4ESMN1; SMN2KMT2A
SCHEMBL6980780 0.73 CACNA2D1 (0.43) GAATSHRTDP1HPGD
Hydrochloric Acid SCHEMBL6984558 0.72 SIGMAR1 (0.43) ALDH1A1POLBSMN1; SMN2MEN1
SCHEMBL6974100 0.72 NPC1 (0.48) ALDH1A1POLBCYP2C19KDM4EMAPT
Hydrochloric Acid SCHEMBL6983896 0.72 SIGMAR1 (0.48) ALDH1A1KDM4EKMT2AGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed