SCHEMBL6984888

SCHEMBL6984888

CN(C(=O)Oc1ccc2c(c1)CCCN2C(=O)CCc1ccc(C(=N)N)cc1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.44
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
MAPK1 P28482 1/20 0.44
HSD17B10 Q99714 1/20 0.41
ALDH1A1 P00352 4/20 0.40
ITGB3 P05106 2/20 0.40
ITGA2B P08514 2/20 0.40
TSHR P16473 2/20 0.39
ACHE P22303 1/20 0.39
LMNA P02545 1/20 0.39
PARP1 P09874 1/20 0.39
MEN1 O00255 1/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 1/20 0.39
ESR1 P03372 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
CHRM1 P11229 1/20 0.39
ADORA1 P30542 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7080783 0.87 POLB (0.48) MAPTNPC1RAB9ASMN1; SMN2MAPK1
SCHEMBL6985405 0.86 HSD17B10 (0.46) MAPTNPC1RAB9ASMN1; SMN2MAPK1
Hydrochloric Acid SCHEMBL6980241 0.86 POLB (0.48) MAPTNPC1RAB9ASMN1; SMN2MAPK1
SCHEMBL6982704 0.83 ITGB3 (0.44) MAPTNPC1RAB9ASMN1; SMN2MAPK1
Hydrochloric Acid SCHEMBL6985632 0.81 ITGB3 (0.41) MAPTNPC1RAB9ASMN1; SMN2MAPK1
SCHEMBL6978012 0.81 NR3C1 (0.49) MAPTALDH1A1LMNAMEN1HPGD
Hydrochloric Acid SCHEMBL6985575 0.81 RXRA (0.48) MAPTNPC1RAB9ASMN1; SMN2MAPK1
Hydrochloric Acid SCHEMBL6982241 0.80 NR3C1 (0.48) MAPTALDH1A1LMNAMEN1HPGD
Hydrochloric Acid SCHEMBL7956681 0.80 NR3C1 (0.42) MAPTNPC1RAB9ASMN1; SMN2MAPK1
SCHEMBL7958817 0.80 NR3C1 (0.47) MAPTALDH1A1LMNAMEN1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed