SCHEMBL6984897

SCHEMBL6984897

Cc1c(C)c2c(c(C)c1N)CC(C)(CN1CCc3ccccc3C1)O2

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 2/20 0.38
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
CXCR3 P49682 1/20 0.35
CD44 P16070 1/20 0.35
GAA P10253 2/20 0.35
MAPT P10636 2/20 0.35
DHFR P00374 1/20 0.34
KDM4E B2RXH2 1/20 0.34
HTT P42858 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
CARM1 Q86X55 1/20 0.34
HTR1A P08908 1/20 0.34
HTR2A P28223 1/20 0.34
HTR7 P34969 1/20 0.34
HTR2B P41595 1/20 0.34
NOS1 P29475 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981092 0.94 DRD3 (0.34) DRD3KMT2AMEN1CXCR3CD44
Oxalic Acid SCHEMBL6978638 0.94 KDM4E (0.41) DRD3KMT2AMEN1GAAMAPT
Hydrochloric Acid SCHEMBL6982794 0.93 KMT2A (0.35) DRD3KMT2AMEN1CXCR3GAA
SCHEMBL3936672 0.80 HTR1A (0.46) KMT2AMEN1GAADHFRKDM4E
SCHEMBL6983488 0.79 DRD2 (0.41) DRD3KMT2AMEN1MAPTKDM4E
SCHEMBL6985365 0.79 LMNA (0.42)
SCHEMBL8718755 0.78 USP2 (0.35) DRD3KMT2AMAPTHTR2B
SCHEMBL8713358 0.78 USP2 (0.38) DRD3KMT2AMAPTHTR2B
Hydrochloric Acid SCHEMBL6979044 0.78 LMNA (0.41) KMT2AMEN1MAPT
SCHEMBL8713753 0.77 USP2 (0.38) DRD3KMT2AMEN1MAPTHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed