SCHEMBL6986313

SCHEMBL6986313

CC1=C(C)C2=C(N)C(C)(CN3CC=C(c4c[nH]c5ccccc45)CC3)CC2=C(C)O1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.53
LMNA P02545 3/20 0.53
ALOX15 P16050 3/20 0.53
HTR1A P08908 10/20 0.49
DRD2 P14416 8/20 0.49
HTR2A P28223 4/20 0.49
HTT P42858 2/20 0.49
SLC6A4 P31645 2/20 0.46
POLB P06746 1/20 0.46
HTR6 P50406 1/20 0.46
HSD17B10 Q99714 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
SIGMAR1 Q99720 1/20 0.43
TDO2 P48775 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6986246 0.79 ADRA1D (0.46) KDM4ESLC6A4POLB
SCHEMBL6986305 0.72 KDM4E (0.53) KDM4ELMNAALOX15HTR1ADRD2
SCHEMBL11321052 0.71 KDM4E (1.00) KDM4ELMNAALOX15HTR1ADRD2
Hydrochloric Acid SCHEMBL11325899 0.71 KDM4E (1.00) KDM4ELMNAALOX15HTR1ADRD2
Hydrochloric Acid SCHEMBL6979051 0.70 LMNA (0.41) KDM4ELMNADRD2HTTPOLB
SCHEMBL11315106 0.69 KDM4E (0.81) KDM4ELMNAALOX15HTR1ADRD2
Hydrochloric Acid SCHEMBL11313113 0.69 KDM4E (0.81) KDM4ELMNAALOX15HTR1ADRD2
SCHEMBL4469442 0.69 KDM4E (0.76) KDM4ELMNAALOX15HTR1ADRD2
Hydrochloric Acid SCHEMBL6985853 0.69 DRD2 (0.40) HTR1ADRD2SIGMAR1
SCHEMBL11314586 0.69 KDM4E (0.71) KDM4ELMNAALOX15HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed