SCHEMBL6986414

SCHEMBL6986414

CC(C)C[C@@H](C(=O)NN(CC(C)C)C(=O)Cn1ccnc1)[C@H](CCNC(=O)c1ccccc1)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 5/20 0.39
NAMPT P43490 7/20 0.36
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6987473 0.90 CYP26A1 (0.39) CYP26A1NAMPTNPC1RAB9ASMN1; SMN2
SCHEMBL6988045 0.89 CYP26A1 (0.38) CYP26A1NAMPTNPC1RAB9ASMN1; SMN2
SCHEMBL6981905 0.85 HRH4 (0.39) CYP26A1NAMPTALDH1A1MAPTTSHR
SCHEMBL6987187 0.75 TBXAS1 (0.41) NAMPTALDH1A1
SCHEMBL6980588 0.74 NPC1 (0.48) NPC1RAB9ASMN1; SMN2
SCHEMBL6980590 0.74 NPC1 (0.48) NPC1RAB9ASMN1; SMN2
SCHEMBL6985273 0.73 ADAM17 (0.59)
SCHEMBL6983142 0.73 NPC1 (0.42) NPC1RAB9ASMN1; SMN2
SCHEMBL6986413 0.70 CYP26A1 (0.37) CYP26A1NAMPTMAPT
SCHEMBL6982700 0.69 MMP1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1089964-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-10-29 EP disclosed
US-6239151-B1 TREATMENT OF INFLAMMATORY AND AUTOIMMUNE DISEASES, OSTEOARTHRITIS, RESPIRATORY DISEASES, TUMORS, CACHEXIA, CARDIOVASCULAR DISEASES, FEVER, HAEMORRHAGE AND SEPSIS, HYDRAZINE DERIVATIVES, HOFFMANN-LA ROCHE INC. 2001-05-29 US disclosed