SCHEMBL6988045

SCHEMBL6988045

CC(C)C[C@@H](C(=O)NN(CC(C)C)C(=O)Cn1ccnc1)[C@H](CCNC(=O)c1ccccc1)C(=O)NO

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 4/20 0.38
ADAM17 P78536 1/20 0.38
NAMPT P43490 1/20 0.37
NPC1 O15118 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
RAB9A P51151 1/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
KMT2A Q03164 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
PTGS2 P35354 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6987473 0.94 CYP26A1 (0.39) CYP26A1NAMPTNPC1SMN1; SMN2RAB9A
SCHEMBL6981905 0.89 HRH4 (0.39) CYP26A1NAMPTNPC1RAB9A
SCHEMBL6986414 0.89 CYP26A1 (0.39) CYP26A1NAMPTNPC1SMN1; SMN2RAB9A
SCHEMBL6987187 0.85 TBXAS1 (0.41) ADAM17NAMPTCYP3A4CYP2D6
SCHEMBL6985273 0.82 ADAM17 (0.59) ADAM17CYP3A4CYP2D6
SCHEMBL6982700 0.79 MMP1 (0.42) CYP3A4CYP2D6
SCHEMBL6981814 0.79 MMP1 (0.42) CYP3A4CYP2D6
SCHEMBL7816201 0.78 MMP1 (0.44) CYP3A4CYP2D6
SCHEMBL6980338 0.74 ADAM17 (0.54) ADAM17CYP3A4CYP2D6
SCHEMBL6984204 0.71 ADAM17 (0.64) ADAM17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1089964-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-10-29 EP disclosed
US-6239151-B1 TREATMENT OF INFLAMMATORY AND AUTOIMMUNE DISEASES, OSTEOARTHRITIS, RESPIRATORY DISEASES, TUMORS, CACHEXIA, CARDIOVASCULAR DISEASES, FEVER, HAEMORRHAGE AND SEPSIS, HYDRAZINE DERIVATIVES, HOFFMANN-LA ROCHE INC. 2001-05-29 US disclosed