SCHEMBL6987649

SCHEMBL6987649

FC(F)(F)c1[c]cccc1-c1ccccc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 4/20 0.41
NOTUM Q6P988 2/20 0.39
CYP3A4 P08684 3/20 0.37
ALOX15 P16050 3/20 0.37
HSD17B10 Q99714 3/20 0.37
CYP1A2 P05177 3/20 0.37
CYP2D6 P10635 3/20 0.37
MAPK1 P28482 2/20 0.37
ALDH1A1 P00352 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
CYP2C19 P33261 2/20 0.37
TSHR P16473 1/20 0.37
HIF1A Q16665 1/20 0.37
HPGD P15428 1/20 0.37
AR P10275 1/20 0.37
TRPA1 O75762 3/20 0.36
SCN9A Q15858 1/20 0.36
PSMB8 P28062 1/20 0.36
CYP2C9 P11712 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL82438 0.81 TDP1 (0.34) HSD11B1NOTUMALDH1A1TDP1
SCHEMBL12817256 0.81 HSD11B1 (0.41) HSD11B1NOTUMCYP3A4ALOX15HSD17B10
SCHEMBL2431241 0.81 HTR1A (0.33) HSD11B1NOTUMALDH1A1
SCHEMBL3416823 0.79 HSD11B1 (0.41) HSD11B1NOTUMCYP3A4ALOX15HSD17B10
SCHEMBL6334156 0.79 AR (0.36) HSD11B1AR
SCHEMBL11032497 0.79 ALDH1A1 (0.38) HSD11B1HSD17B10MAPK1ALDH1A1
SCHEMBL3583635 0.79 CYP2A6 (0.38) HSD11B1ALDH1A1TSHRHPGDAR
SCHEMBL455371 0.78 ALDH1A1 (0.40) HSD11B1HSD17B10MAPK1ALDH1A1TSHR
SCHEMBL197671 0.78 HSD11B1 (0.56) HSD11B1NOTUMCYP3A4ALOX15HSD17B10
SCHEMBL3636361 0.78 HSD11B1 (0.42) HSD11B1NOTUMCYP3A4ALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0937051-A1 FUNGICIDAL CYCLIC AMIDES E.I. DU PONT DE NEMOURS & COMPANY INCORPORATED (US) 1999-08-25 EP claimed
WO-1998020003-A1 FUNGICIDAL CYCLIC AMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-05-14 WO claimed
EP-1318984-A1 4-AMINO-QUINAZOLINES MERCK PATENT GmbH (DE) 2003-06-18 EP disclosed
WO-2002024667-A1 4-AMINO-QUINAZOLINES MERCK PATENT GMBH (DE) 2002-03-28 WO disclosed