SCHEMBL11032497

SCHEMBL11032497

FC(F)(F)c1[c]cccc1-c1ccccc1Br

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
MAPK1 P28482 1/20 0.38
HSD11B1 P28845 1/20 0.37
TACR1 P25103 1/20 0.35
PDK2 Q15119 1/20 0.33
IDO1 P14902 1/20 0.33
LMNA P02545 1/20 0.33
ACHE P22303 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PBRM1 Q86U86 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA5A P35218 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9770289 0.86 ENPP3 (0.33) PDK2
SCHEMBL28126011 0.83 PTPRC (0.36) MAPK1PDK2
SCHEMBL1068615 0.82 ENPP3 (0.33) CA1CA2CA5ACA9
SCHEMBL28839943 0.80 PDK2 (0.35) HSD11B1PDK2
SCHEMBL6987649 0.79 HSD11B1 (0.41) ALDH1A1MAPK1HSD11B1HSD17B10
SCHEMBL2431241 0.79 HTR1A (0.33) ALDH1A1HSD11B1PDK2IDO1
SCHEMBL6334156 0.78 AR (0.36) HSD11B1TACR1PDK2
SCHEMBL3583635 0.78 CYP2A6 (0.38) ALDH1A1HSD11B1TACR1PDK2LMNA
SCHEMBL15637106 0.77 CDC25B (0.36) HSD11B1PDK2
SCHEMBL455371 0.77 ALDH1A1 (0.40) ALDH1A1MAPK1HSD11B1TACR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3126335-A1 N-(1-(HETERO)ARYL-1H-PYRAZOL-4-YL)-(HETERO)ARYLAMIDE DERIVATIVES AND USE THEREOF AS PESTICIDES Bayer CropScience Aktiengesellschaft (DE) 2017-02-08 EP disclosed
WO-2015150300-A1 N-(1-(HETERO)ARYL-1H-PYRAZOL-4-YL)-(HETERO)ARYLAMIDE DERIVATIVES AND USE THEREOF AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2015-10-08 WO disclosed
EP-2903440-A1 HETEROCYCLIC COMPOUNDS AS PESTICIDES Bayer CropScience AG (DE) 2015-08-12 EP disclosed
WO-2014053450-A1 HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2014-04-10 WO disclosed
US-4455421-A ANTIFERTILITY, ANTIULCER AGENTS; TETRAZOLE DERIVATIVES PFIZER INC. (US) 1984-06-19 US disclosed
US-4365077-A ANTIFERTILITY, ANTIULCER PFIZER INC. (US) 1982-12-21 US disclosed
US-4277484-A ANTIINFLAMMATORY AGENTS CIBA-GEIGY CORPORATION (US) 1981-07-07 US disclosed
US-4157341-A 11-Desoxy-16-aryloxy-ω-tetranorprostaglandins PFIZER INC. (US) 1979-06-05 US disclosed