SCHEMBL6988752

SCHEMBL6988752

COc1c(NCC(=O)NCC2CCN(C3CCCC3)CC2)cccc1C(=O)c1ccc2cc[nH]c2c1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 2/20 0.43
MAPT P10636 2/20 0.43
HPGD P15428 2/20 0.43
HSD17B10 Q99714 2/20 0.43
CHRM2 P08172 2/20 0.39
F10 P00742 5/20 0.38
ALOX12 P18054 1/20 0.37
HTR4 Q13639 1/20 0.36
SMYD3 Q9H7B4 1/20 0.35
JAK2 O60674 1/20 0.35
GHSR Q92847 1/20 0.35
CCR3 P51677 2/20 0.35
SIGMAR1 Q99720 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985512 0.88 KDM4E (0.45) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL7098081 0.79 ACHE (0.41) ALDH1A1KDM4EMAPTHPGDHSD17B10
Hydrochloric Acid SCHEMBL7140810 0.79 ACHE (0.41) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL6986644 0.77 F10 (0.43) ALDH1A1CHRM2F10
SCHEMBL5868270 0.73 ALDH1A1 (0.44) ALDH1A1KDM4EMAPTHPGDHSD17B10
Hydrochloric Acid SCHEMBL6984942 0.73 ROCK2 (0.42) ALDH1A1MAPTF10HTR4
SCHEMBL6989025 0.73 HTR4 (0.43) ALDH1A1HTR4
SCHEMBL5868023 0.71 KDM4E (0.48) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL6987891 0.71 F10 (0.38) ALDH1A1KDM4EF10CCR3
SCHEMBL5868145 0.70 ALDH1A1 (0.50) ALDH1A1KDM4EMAPTHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289954-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2003-03-12 EP disclosed
WO-2001096303-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2001-12-20 WO disclosed