SCHEMBL6989882

SCHEMBL6989882

COc1ccccc1N1CCN(CCCCCn2ccc3c2C(=O)N(Cc2ccccc2)CCC3=O)CC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 11/20 0.57
DRD2 P14416 11/20 0.57
DRD1 P21728 2/20 0.57
DRD4 P21917 5/20 0.55
HTR7 P34969 5/20 0.53
HTR1A P08908 4/20 0.53
ALDH1A1 P00352 2/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
ALOX12 P18054 1/20 0.53
ADRA1D P25100 1/20 0.53
ADRA1A P35348 1/20 0.53
ADRA1B P35368 1/20 0.53
HIF1A Q16665 1/20 0.53
HSD17B10 Q99714 1/20 0.53
KDM4E B2RXH2 1/20 0.52
GLA P06280 1/20 0.52
HPGD P15428 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6989466 0.87 HTR1A (0.59) DRD3DRD2DRD1DRD4HTR7
SCHEMBL6984158 0.86 HTR1A (0.60) DRD3DRD2DRD1DRD4HTR7
SCHEMBL6988196 0.85 HTR1A (0.50) DRD3DRD2HTR7HTR1AHTR6
SCHEMBL6991218 0.85 HTR1A (0.50) DRD3DRD2HTR7HTR1AHTR6
SCHEMBL6984315 0.84 HTR1A (0.49) DRD3DRD2DRD4HTR7HTR1A
SCHEMBL6990381 0.82 HTR1A (0.49) DRD3DRD2DRD4HTR7HTR1A
SCHEMBL6990417 0.81 DRD3 (0.67) DRD3DRD2DRD1DRD4HTR7
SCHEMBL6990656 0.79 ADRA1D (0.47) DRD3DRD2DRD4HTR7HTR1A
SCHEMBL6987269 0.78 L3MBTL1 (0.38) HTR7HTR1AMEN1KMT2A
SCHEMBL6986608 0.78 L3MBTL1 (0.38) HTR7HTR1AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0551527-B1 PYRROLOAZEPINE DERIVATIVE SUNTORY LTD (JP) 2003-04-02 EP disclosed
US-5397780-A Antiserotonine, hypotensive, congestive heart failure SUNTORY LIMITED (JP) 1995-03-14 US disclosed
EP-0551527-A1 PYRROLOAZEPINE DERIVATIVE SUNTORY LIMITED (JP) 1993-07-21 EP disclosed