SCHEMBL6990486

SCHEMBL6990486

CN(CCc1cccc(Cl)c1)C(=O)c1nc2ccccc2nc1O

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.48
AOC3 Q16853 1/20 0.46
PIN1 Q13526 1/20 0.43
CCKAR P32238 1/20 0.42
CCKBR P32239 1/20 0.42
OXTR P30559 1/20 0.41
CSNK1D P48730 1/20 0.41
NPC1 O15118 1/20 0.40
MEN1 O00255 1/20 0.39
HCRTR1 O43613 1/20 0.39
KMT2A Q03164 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
MLYCD O95822 1/20 0.39
RIPK1 Q13546 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6991167 0.88 PIN1 (0.52) AOC3PIN1NPC1MEN1KMT2A
SCHEMBL6987408 0.86 MLYCD (0.51) MLYCD
SCHEMBL6989696 0.80 NPC1 (0.55) NPC1MEN1KMT2AKDM4E
SCHEMBL6990995 0.76 KMT2A (0.54) PIN1MEN1KMT2A
SCHEMBL6989375 0.75 KMT2A (0.50) NPC1MEN1KMT2AKDM4EMAPT
SCHEMBL8242118 0.72 MEN1 (0.57) TAAR1AOC3MEN1KMT2AHPGD
SCHEMBL6989399 0.71 ALDH1A1 (0.40) KMT2AKDM4EMAPT
SCHEMBL6989665 0.69 NPC1 (0.40) NPC1MAPT
SCHEMBL19616099 0.68 L3MBTL1 (0.51) TAAR1AOC3MEN1KMT2AMLYCD
SCHEMBL3056908 0.67 TAAR1 (1.00) TAAR1AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8889683-B2 Substituted quinoxalines as inhibitors of fatty acid binding protein MERCK SHARP & DOHME CORP. (US) 2014-11-18 US disclosed
US-8889683-B2 Substituted quinoxalines as inhibitors of fatty acid binding protein MERCK SHARP & DOHME CORP. (US) 2014-11-18 US disclosed
US-20120122837-A1 INHIBITORS OF FATTY ACID BINDING PROTEIN MERCK SHARP & DOHME LLC 2012-05-17 US disclosed
US-20120122837-A1 INHIBITORS OF FATTY ACID BINDING PROTEIN MERCK SHARP & DOHME LLC 2012-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120122837-A1 INHIBITORS OF FATTY ACID BINDING PROTEIN FABP4, FABP1, FABP3 TAAR1 4179/4885AOC3 4668/4885PIN1 1158/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.