SCHEMBL6990762

SCHEMBL6990762

CSc1cccc2[nH]c(C#N)c(-c3ccc(NC(=O)c4cccnc4)cc3)c12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.56
KMT2A Q03164 2/20 0.56
MEN1 O00255 1/20 0.56
POLB P06746 1/20 0.56
ALOX15 P16050 1/20 0.48
HTT P42858 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
RAB9A P51151 5/20 0.46
GAA P10253 2/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
NPC1 O15118 3/20 0.46
MAPT P10636 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
GFER P55789 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
TP53 P04637 2/20 0.43
ROCK2 O75116 1/20 0.43
ROCK1 Q13464 1/20 0.43
LMNA P02545 2/20 0.41
HIF1A Q16665 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6986415 0.74 RAB9A (0.52) ALDH1A1KMT2AMEN1POLBALOX15
SCHEMBL6991349 0.72 SMN1; SMN2 (0.52) KMT2AMEN1POLBHTTRAB9A
SCHEMBL6988214 0.70 GAK (0.49) ALDH1A1KMT2AMEN1POLBHTT
SCHEMBL7141571 0.70 ALDH1A1 (0.59) ALDH1A1KMT2AMEN1POLBALOX15
SCHEMBL22983039 0.69 CYP11B1 (0.74) ALDH1A1KMT2AMEN1POLBRAB9A
SCHEMBL7701971 0.68 MEN1 (0.45) KMT2AMEN1HTTL3MBTL1RAB9A
SCHEMBL2339343 0.67 ALDH1A1 (1.00) ALDH1A1KMT2AMEN1POLBALOX15
SCHEMBL27754792 0.66 ROCK2 (0.66) ALDH1A1KMT2AMEN1RAB9AGAA
SCHEMBL1971026 0.65 NAMPT (0.78) ALDH1A1KMT2AHTTRAB9AGAA
SCHEMBL8252721 0.65 RAB9A (1.00) ALDH1A1KMT2APOLBRAB9AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303508-A1 SUBSTITUTED 1-(4-AMINOPHENYL)INDOLES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2003-04-23 EP disclosed
WO-2002006273-A1 SUBSTITUTED 1-(4-AMINOPHENYL)INDOLES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-01-24 WO disclosed