SCHEMBL6990778

SCHEMBL6990778

NS(=O)(=O)c1ccc(NC(=O)O)cc1

nearest known ligand 0.74

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.74
CA1 P00915 14/20 0.70
CA2 P00918 14/20 0.70
CA12 O43570 12/20 0.70
CA9 Q16790 12/20 0.70
PTPN7 P35236 2/20 0.68
CA4 P22748 2/20 0.64
CA14 Q9ULX7 2/20 0.64
CA7 P43166 2/20 0.62
MEN1 O00255 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28499329 0.85 KMT2A (1.00) KMT2ACA1CA2CA12CA9
SCHEMBL358576 0.83 CA1 (0.80) KMT2ACA1CA2CA12CA9
SCHEMBL671546 0.82 CA2 (1.00) KMT2ACA1CA2CA12CA9
SCHEMBL29941244 0.82 PTPN7 (0.71) KMT2ACA1CA2CA12CA9
Acetylsulfanilamide SCHEMBL359721 0.82 CA1 (1.00) KMT2ACA1CA2CA12CA9
SCHEMBL9280164 0.81 PTPN7 (1.00) KMT2ACA1CA2CA12CA9
Bicarbonate SCHEMBL5658794 0.81 KMT2A (0.65) KMT2ACA1CA2CA12CA9
SCHEMBL10458764 0.81 TIMP3 (0.54) KMT2ACA1CA2CA12CA9
Acetylsulfanilamide SCHEMBL8043497 0.80 CA1 (0.96) KMT2ACA1CA2CA12CA9
SCHEMBL9130898 0.80 GAA (0.68) KMT2ACA1CA2CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180339963-A1 ANTICONVULSANT CARBAMATE DERIVATIVES YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD. (IL) 2018-11-29 US claimed
WO-1997027226-A2 HIGHLY FUNCTIONALIZED POLYETHYLENE GLYCOL GRAFTED POLYSTYRENE SUPPORTS ARGONAUT TECHNOLOGIES, INC. (US) 1997-07-31 WO claimed
US-20180339963-A1 ANTICONVULSANT CARBAMATE DERIVATIVES YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD. (IL) 2018-11-29 US disclosed
CN-101472925-B As adenosine A2APurine derivatives of receptor agonists NOVARTIS AG 2012-06-13 CN disclosed
CN-101479267-B Purine derivatives as A2A agonists NOVARTIS AG 2012-05-02 CN disclosed
CN-101479267-A Purine derivatives as A2A agonists NOVARTIS AG (CH) 2009-07-08 CN disclosed
CN-101472925-A As adenosine A2APurine derivatives of receptor agonists NOVARTIS AG (CH) 2009-07-01 CN disclosed
EP-0874809-B1 CARBAMOYLOXY DERIVATIVES OF MUTILINE AND THEIR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2003-08-27 EP disclosed
US-6239175-B1 Carbamoyloxy derivatives of mutiline and their use as antibacterials SMITHKLINE BEECHAM P.L.C. (GB) 2001-05-29 US disclosed
US-6020368-A MICROBIOCIDES HINKS JEREMY DAVID (US) 2000-02-01 US disclosed
EP-0874809-A1 CARBAMOYLOXY DERIVATIVES OF MUTILINE AND THEIR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 1998-11-04 EP disclosed
CN-1036395-C Piperazine derivatives WYETH JOHN & BROTHER LTD (GB) 1997-11-12 CN disclosed
WO-1997027226-A2 HIGHLY FUNCTIONALIZED POLYETHYLENE GLYCOL GRAFTED POLYSTYRENE SUPPORTS ARGONAUT TECHNOLOGIES, INC. (US) 1997-07-31 WO disclosed
WO-1997025309-A1 CARBAMOYLOXY DERIVATIVES OF MUTILINE AND THEIR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 1997-07-17 WO disclosed
CN-1076446-A Bridged piperazine derivatives WYETH JOHN & BROTHER LTD (GB) 1993-09-22 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180339963-A1 ANTICONVULSANT CARBAMATE DERIVATIVES CNR2, GRIK5, GRIK4 KMT2A 318/4885CA1 22/4885CA2 46/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.