SCHEMBL6991739

SCHEMBL6991739

O=C(NCC(C(=O)NC12CCCC1OCC2=O)c1ccc(Cl)cc1)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 5/20 0.38
TP53 P04637 3/20 0.37
GCGR P47871 5/20 0.37
GIPR P48546 2/20 0.37
LMNA P02545 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
CTSS P25774 1/20 0.35
SCN8A Q9UQD0 1/20 0.35
PREP P48147 1/20 0.35
LIPE Q05469 1/20 0.35
SCN9A Q15858 1/20 0.35
ADCY6 O43306 1/20 0.35
ADCY3 O60266 1/20 0.35
ADCY9 O60503 1/20 0.35
ADCY5 O95622 1/20 0.35
ADCY8 P40145 1/20 0.35
ADCY7 P51828 1/20 0.35
ADCY2 Q08462 1/20 0.35
ADCY1 Q08828 1/20 0.35
ADCY4 Q8NFM4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6992582 0.94 TRPV1 (0.36) TRPV1GCGRCTSSPREPSCN9A
SCHEMBL6998484 0.93 TRPV1 (0.39) TRPV1GCGRPREPSCN9AADCY6
SCHEMBL7144829 0.92 TRPV1 (0.42) TRPV1GCGRPTGDR2PREPSCN9A
SCHEMBL6988915 0.90 IDO1 (0.42) TP53LMNAPTGDR2
SCHEMBL6994067 0.88 RAB9A (0.41) TP53LMNAPTGDR2
SCHEMBL6989614 0.87 TP53 (0.47) TP53GCGRLMNAADCY6ADCY3
SCHEMBL6988021 0.85 NPC1 (0.39) TP53LMNA
SCHEMBL6988551 0.84 TP53 (0.35) TP53GCGRGIPR
SCHEMBL6997966 0.83 MEN1 (0.34) GCGRGIPR
SCHEMBL6699086 0.83 KLKB1 (0.43) GCGRGIPRCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358176-A2 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES Amura Therapeutics Limited (GB) 2003-11-05 EP disclosed
WO-2002057246-A2 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES AMURA THERAPEUTICS LIMITED (GB) 2002-07-25 WO disclosed