SCHEMBL6992582

SCHEMBL6992582

O=C(NCC(C(=O)NC12CCCC1OCC2=O)c1ccc(F)cc1)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 7/20 0.36
PREP P48147 1/20 0.36
SCN9A Q15858 1/20 0.36
GCGR P47871 3/20 0.36
ADCY6 O43306 1/20 0.36
ADCY3 O60266 1/20 0.36
ADCY9 O60503 1/20 0.36
ADCY5 O95622 1/20 0.36
ADCY8 P40145 1/20 0.36
ADCY7 P51828 1/20 0.36
ADCY2 Q08462 1/20 0.36
ADCY1 Q08828 1/20 0.36
ADCY4 Q8NFM4 1/20 0.36
CTSL P07711 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
TAOK1 Q7L7X3 1/20 0.35
TAOK3 Q9H2K8 1/20 0.35
SLC6A9 P48067 1/20 0.34
EPHX2 P34913 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6998484 0.94 TRPV1 (0.39) TRPV1PREPSCN9AGCGRADCY6
SCHEMBL6991739 0.94 TRPV1 (0.38) TRPV1PREPSCN9AGCGRADCY6
SCHEMBL6988551 0.90 TP53 (0.35) GCGRSLC6A9
SCHEMBL7144829 0.90 TRPV1 (0.42) TRPV1PREPSCN9AGCGRTAOK1
SCHEMBL6997966 0.84 MEN1 (0.34) GCGRPDE2A
SCHEMBL6988915 0.83 IDO1 (0.42)
SCHEMBL6992575 0.82 USP30 (0.48) SCN9ACTSLCTSSCTSKEPHX2
SCHEMBL6294364 0.81 TP53 (0.38) GCGRADCY6ADCY3ADCY9ADCY5
SCHEMBL6988745 0.81 CTSK (0.35) CTSK
SCHEMBL6994067 0.81 RAB9A (0.41) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358176-A2 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES Amura Therapeutics Limited (GB) 2003-11-05 EP disclosed
WO-2002057246-A2 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES AMURA THERAPEUTICS LIMITED (GB) 2002-07-25 WO disclosed