SCHEMBL6988915

SCHEMBL6988915

O=C(NCC(C(=O)NC12CCCC1OCC2=O)c1ccc(Cl)cc1)c1ccc(OC(F)F)cc1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.42
KMT2A Q03164 2/20 0.40
TP53 P04637 5/20 0.39
LMNA P02545 1/20 0.39
PTGDR2 Q9Y5Y4 5/20 0.38
ATM Q13315 1/20 0.36
THRB P10828 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
MDM2 Q00987 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6993342 0.93 KMT2A (0.40) IDO1KMT2ATP53LMNAPTGDR2
SCHEMBL6991739 0.90 TRPV1 (0.38) TP53LMNAPTGDR2
SCHEMBL6994067 0.88 RAB9A (0.41) IDO1KMT2ATP53LMNAPTGDR2
SCHEMBL6990244 0.88 TP53 (0.38) IDO1KMT2ATP53PTGDR2THRB
SCHEMBL6989614 0.86 TP53 (0.47) KMT2ATP53LMNATHRBSMN1; SMN2
SCHEMBL6988021 0.85 NPC1 (0.39) KMT2ATP53LMNATHRBSMN1; SMN2
SCHEMBL6992582 0.83 TRPV1 (0.36)
SCHEMBL6998484 0.82 TRPV1 (0.39)
SCHEMBL6300424 0.82 IDO1 (0.44) IDO1KMT2ASMN1; SMN2
SCHEMBL6988745 0.82 CTSK (0.35) KMT2ALMNASMN1; SMN2NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358176-A2 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES Amura Therapeutics Limited (GB) 2003-11-05 EP disclosed
WO-2002057246-A2 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES AMURA THERAPEUTICS LIMITED (GB) 2002-07-25 WO disclosed