SCHEMBL6991977

SCHEMBL6991977

O=C(O)NC(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.59
CES1 P23141 1/20 0.59
NPC1 O15118 2/20 0.57
RAB9A P51151 2/20 0.57
CRHBP P24387 1/20 0.57
CRHR2 Q13324 1/20 0.57
SRD5A2 P31213 1/20 0.57
PTPN1 P18031 2/20 0.55
TRPV1 Q8NER1 2/20 0.51
PTGS1 P23219 2/20 0.51
GSK3B P49841 2/20 0.50
KDM4E B2RXH2 1/20 0.50
APAF1 O14727 1/20 0.50
TDP2 O95551 1/20 0.50
NSD2 O96028 1/20 0.50
MAPT P10636 1/20 0.50
CASP3 P42574 1/20 0.50
GALK1 P51570 1/20 0.50
BLM P54132 1/20 0.50
KMT2A Q03164 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31433394 0.84 ALDH1A1 (0.50) NPC1RAB9AMAPTKMT2A
SCHEMBL26163219 0.82 CES2 (0.57) CES2CES1NPC1RAB9ACRHBP
SCHEMBL25142228 0.82 CES2 (0.57) CES2CES1NPC1RAB9ACRHBP
SCHEMBL15328058 0.82 PTGS1 (0.59) CES2CES1NPC1RAB9ACRHBP
SCHEMBL24534899 0.81 PTPN1 (0.53) CES2CES1NPC1RAB9ACRHBP
SCHEMBL3655196 0.81 CES2 (0.61) CES2CES1NPC1RAB9ACRHBP
SCHEMBL6991713 0.80 LMNA (0.67) CES2RAB9ASRD5A2PTGS1MAPT
Benzene SCHEMBL28007806 0.79 KMT2A (0.56) NPC1RAB9ACRHBPCRHR2PTPN1
SCHEMBL3418657 0.79 CES2 (0.53) CES2CES1NPC1RAB9ACRHBP
SCHEMBL14880225 0.78 CES2 (0.64) CES2CES1SRD5A2TRPV1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0874809-B1 CARBAMOYLOXY DERIVATIVES OF MUTILINE AND THEIR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2003-08-27 EP claimed
US-6239175-B1 Carbamoyloxy derivatives of mutiline and their use as antibacterials SMITHKLINE BEECHAM P.L.C. (GB) 2001-05-29 US claimed
EP-0874809-B1 CARBAMOYLOXY DERIVATIVES OF MUTILINE AND THEIR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2003-08-27 EP disclosed
US-6239175-B1 Carbamoyloxy derivatives of mutiline and their use as antibacterials SMITHKLINE BEECHAM P.L.C. (GB) 2001-05-29 US disclosed
US-6020368-A MICROBIOCIDES HINKS JEREMY DAVID (US) 2000-02-01 US disclosed