SCHEMBL6992649

SCHEMBL6992649

Nc1cc(-c2ccc3ccccc3c2)[nH]n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
KMT2A Q03164 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
MKNK1 Q9BUB5 1/20 0.56
MKNK2 Q9HBH9 1/20 0.56
MEN1 O00255 1/20 0.56
USP2 O75604 1/20 0.56
DYRK1A Q13627 1/20 0.56
CYP11B1 P15538 1/20 0.53
CYP11B2 P19099 1/20 0.53
MITF O75030 1/20 0.51
TP53 P04637 1/20 0.51
IKBKB O14920 1/20 0.51
LTA4H P09960 1/20 0.51
LMNA P02545 1/20 0.49
NPC1 O15118 2/20 0.49
MAPT P10636 2/20 0.49
RAB9A P51151 2/20 0.49
GFER P55789 2/20 0.49
CYP1A2 P05177 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2089082 0.80 DYRK1A (0.77) ALDH1A1KMT2ASMN1; SMN2MKNK1MKNK2
SCHEMBL6956022 0.79 ALDH1A1 (0.67) ALDH1A1KMT2ASMN1; SMN2MKNK1MKNK2
SCHEMBL330565 0.79 ALDH1A1 (0.66) ALDH1A1KMT2ASMN1; SMN2MKNK1MKNK2
SCHEMBL4895088 0.79 IKBKB (0.51) ALDH1A1SMN1; SMN2CYP11B1CYP11B2IKBKB
SCHEMBL2662870 0.77 RAB9A (0.70) KMT2ASMN1; SMN2MEN1TP53LMNA
SCHEMBL14190747 0.76 LTA4H (0.74) ALDH1A1KMT2ASMN1; SMN2MKNK1MKNK2
SCHEMBL17279987 0.76 RAB9A (0.58) KMT2ASMN1; SMN2CYP11B1CYP11B2TP53
SCHEMBL26108551 0.75 KDM4E (0.65) ALDH1A1KMT2ASMN1; SMN2MEN1TP53
SCHEMBL28573902 0.75 ALDH1A1 (0.71) ALDH1A1KMT2ASMN1; SMN2MKNK1MKNK2
SCHEMBL3517442 0.73 CA12 (0.56) KMT2AMEN1CYP11B1CYP11B2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945438-B1 PYRAZOLE DERIVATIVES BANYU PHARMA CO LTD (JP) 2003-03-05 EP disclosed
US-6057335-A Pyrazole derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 2000-05-02 US disclosed
EP-0945438-A1 PYRAZOLE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1999-09-29 EP disclosed