SCHEMBL6992679

SCHEMBL6992679

CCN1CCc2sc3ncn(CCCN4CCN(c5ncccn5)CC4)c(=O)c3c2C1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 20/20 0.49
ADRA1D P25100 19/20 0.49
HTR1B P28222 19/20 0.49
ADRA1A P35348 19/20 0.49
ADRA1B P35368 19/20 0.49
HTR7 P34969 3/20 0.48
DRD2 P14416 2/20 0.48
HTR2A P28223 2/20 0.48
DRD3 P35462 2/20 0.48
HTR2C P28335 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6996817 0.94 HTR1A (0.55) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7676469 0.93 HTR1A (0.51) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7676809 0.87 HTR1A (0.56) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL6992475 0.85 HTR1A (0.66) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL6994547 0.85 HTR1A (0.57) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7718492 0.83 HTR1A (0.66) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL6999826 0.81 SIGMAR1 (0.49) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL6999544 0.80 NPC1 (0.60) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL3457893 0.80 SIGMAR1 (0.49) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL6997759 0.80 HTR1A (0.75) HTR1AADRA1DHTR1BADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1023296-B1 3-SUBSTITUTED PYRIDO 3',4':4,5] THIENO 2,3-D] PYRIMIDINE DERIVATIVES, AND PRODUCTION AND USE OF THE SAME ABBOTT GMBH & CO KG (DE) 2003-12-17 EP disclosed
US-6387912-B1 STROKE THERAPY BASF AKTIENGESELLSCHAFT (DE) 2002-05-14 US disclosed
US-6159981-A 3-substituted pyrido [3',4':4,5] Thieno [2,3-d] pyrimidine derivatives, and production and use of the same BASF AKTIENGESELLSCHAFT (DE) 2000-12-12 US disclosed