SCHEMBL6999544

SCHEMBL6999544

CCN1CCc2sc3ncn(CCO)c(=O)c3c2C1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.60
RAB9A P51151 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
SIGMAR1 Q99720 2/20 0.49
POLB P06746 1/20 0.47
ESR2 Q92731 1/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
HTR1A P08908 8/20 0.45
ADRA1D P25100 8/20 0.45
HTR1B P28222 8/20 0.45
ADRA1A P35348 8/20 0.45
ADRA1B P35368 8/20 0.45
P2RX3 P56373 5/20 0.45
RXFP1 Q9HBX9 1/20 0.44
DRD2 P14416 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR7 P34969 1/20 0.42
DRD3 P35462 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3457893 0.89 SIGMAR1 (0.49) NPC1RAB9ASMN1; SMN2SIGMAR1POLB
SCHEMBL6996817 0.82 HTR1A (0.55) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL3457233 0.81 NPC1 (0.67) NPC1RAB9ASMN1; SMN2HTR1AADRA1D
SCHEMBL6992679 0.80 HTR1A (0.49) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7522252 0.80 ALDH1A1 (0.71) NPC1RAB9ASMN1; SMN2POLBESR2
SCHEMBL6994547 0.80 HTR1A (0.57) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL6997759 0.79 HTR1A (0.75) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7001787 0.79 HTR1A (0.75) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL6999826 0.78 SIGMAR1 (0.49) NPC1RAB9ASMN1; SMN2SIGMAR1HTR1A
SCHEMBL6999663 0.78 HTR1A (0.77) HTR1AADRA1DHTR1BADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1023296-B1 3-SUBSTITUTED PYRIDO 3',4':4,5] THIENO 2,3-D] PYRIMIDINE DERIVATIVES, AND PRODUCTION AND USE OF THE SAME ABBOTT GMBH & CO KG (DE) 2003-12-17 EP disclosed
US-6387912-B1 STROKE THERAPY BASF AKTIENGESELLSCHAFT (DE) 2002-05-14 US disclosed
US-6355647-B1 INHIBIT THE SEROTONIN REUPTAKE. HYPERPROLACTINEMIA, VASOSPASMS, HYPERTENSION, GASTROINTESTINAL DISORDERS ASSOCIATED WITH MOTILITY AND SECRETION ABBOTT LABORATORIES 2002-03-12 US disclosed
US-6159981-A 3-substituted pyrido [3',4':4,5] Thieno [2,3-d] pyrimidine derivatives, and production and use of the same BASF AKTIENGESELLSCHAFT (DE) 2000-12-12 US disclosed