SCHEMBL6995228

SCHEMBL6995228

Cc1cc(F)ccc1C(=O)Nc1ccc(C(=O)N2CCCC(=O)c3sccc32)cc1Cl

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 10/20 0.51
AVPR1A P37288 9/20 0.51
AVPR1B P47901 4/20 0.44
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
PYGL P06737 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
MAP3K7 O43318 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6987523 0.94 AVPR2 (0.56) AVPR2AVPR1AAVPR1BNPC1RAB9A
SCHEMBL6991988 0.90 AVPR1A (0.56) AVPR2AVPR1AAVPR1B
SCHEMBL6994183 0.87 AVPR2 (0.60) AVPR2AVPR1AAVPR1B
SCHEMBL6985550 0.87 AVPR2 (0.47) AVPR2AVPR1AAVPR1BMAP3K7
SCHEMBL6989537 0.86 AVPR1A (0.55) AVPR2AVPR1AAVPR1BNPC1RAB9A
SCHEMBL6996850 0.82 LMNA (0.51) AVPR2AVPR1AAVPR1B
SCHEMBL6989178 0.81 AVPR2 (0.69) AVPR2AVPR1AAVPR1B
SCHEMBL6988903 0.77 AVPR2 (0.55) AVPR2AVPR1AAVPR1BHDAC1HDAC6
SCHEMBL6990759 0.75 AVPR1A (0.68) AVPR2AVPR1AAVPR1B
SCHEMBL5321445 0.75 AVPR1A (0.75) AVPR2AVPR1AAVPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0811008-B1 BICYCLIC BENZAZEPINE DERIVATIVES AS VASOPRESSIN ANTAGONISTS WYETH CORP (US) 2003-10-01 EP disclosed