SCHEMBL6997537

SCHEMBL6997537

COc1cccc(C(=O)N=C=O)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.61
CES1 P23141 1/20 0.61
PARP1 P09874 1/20 0.57
NPC1 O15118 7/20 0.53
RAB9A P51151 7/20 0.53
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.49
LMNA P02545 1/20 0.49
ABCG2 Q9UNQ0 1/20 0.49
ESR1 P03372 1/20 0.49
ESR2 Q92731 1/20 0.49
PRSS1 P07477 1/20 0.49
PRSS2 P07478 1/20 0.49
PRSS3 P35030 1/20 0.49
NPSR1 Q6W5P4 2/20 0.48
ALDH1A1 P00352 2/20 0.48
MAPT P10636 1/20 0.48
PKM P14618 1/20 0.48
XBP1 P17861 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5824521 0.85 CES2 (0.59) CES2CES1PARP1NPC1RAB9A
SCHEMBL3887425 0.83 CES2 (0.56) CES2CES1PARP1NPC1RAB9A
SCHEMBL3395919 0.82 L3MBTL1 (0.43) CES2CES1PARP1MEN1KMT2A
SCHEMBL10978364 0.81 CES2 (0.67) CES2CES1PARP1NPC1RAB9A
SCHEMBL27511887 0.80 LOXL2 (0.49) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL18311274 0.79 CES2 (0.65) CES2CES1PARP1NPC1RAB9A
SCHEMBL4246590 0.79 CES2 (0.55) CES2CES1PARP1RAB9AMEN1
Butanedione SCHEMBL28856348 0.79 FURIN (0.38) CES2CES1PARP1NPC1RAB9A
SCHEMBL5555845 0.78 TDP1 (0.40) CES2CES1RAB9AMEN1KMT2A
SCHEMBL4092403 0.77 PARP1 (0.53) PARP1NPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0874809-B1 CARBAMOYLOXY DERIVATIVES OF MUTILINE AND THEIR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2003-08-27 EP disclosed
US-6239175-B1 Carbamoyloxy derivatives of mutiline and their use as antibacterials SMITHKLINE BEECHAM P.L.C. (GB) 2001-05-29 US disclosed
US-6020368-A MICROBIOCIDES HINKS JEREMY DAVID (US) 2000-02-01 US disclosed
EP-0874809-A1 CARBAMOYLOXY DERIVATIVES OF MUTILINE AND THEIR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 1998-11-04 EP disclosed
WO-1997025309-A1 CARBAMOYLOXY DERIVATIVES OF MUTILINE AND THEIR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 1997-07-17 WO disclosed