SCHEMBL7002086

SCHEMBL7002086

NCc1onc2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.42
CYP1A2 P05177 3/20 0.37
SCN8A Q9UQD0 1/20 0.37
IDO1 P14902 1/20 0.37
GPR3 P46089 1/20 0.36
ALDH1A1 P00352 3/20 0.35
HPGD P15428 3/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
KDM4E B2RXH2 2/20 0.35
GLA P06280 2/20 0.35
CASP1 P29466 2/20 0.35
CASP7 P55210 2/20 0.35
HSD17B10 Q99714 2/20 0.35
CHRM2 P08172 1/20 0.35
ADRA2A P08913 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
CHRM1 P11229 1/20 0.35
NQO2 P16083 1/20 0.35
MAOA P21397 1/20 0.35
DRD1 P21728 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11919171 0.79 PTGS1 (0.46) CYP1A2IDO1GPR3ALDH1A1HPGD
SCHEMBL5044710 0.79 ELANE (0.41) LOXL2CYP1A2IDO1GPR3ALDH1A1
SCHEMBL8772908 0.76 ALDH1A1 (0.37) IDO1GPR3ALDH1A1HPGDSMN1; SMN2
SCHEMBL2920597 0.76 CA2 (0.54) IDO1GPR3ALDH1A1HPGDSMN1; SMN2
SCHEMBL8772757 0.75 ALDH1A1 (0.37) IDO1GPR3ALDH1A1HPGDSMN1; SMN2
SCHEMBL1027461 0.73 SMN1; SMN2 (0.43) ALDH1A1HPGDSMN1; SMN2KDM4EGLA
SCHEMBL2493164 0.73 PARP1 (0.43) CYP1A2ALDH1A1HPGDSMN1; SMN2KDM4E
SCHEMBL3229873 0.73 LMNA (0.40) CYP1A2GPR3ALDH1A1SMN1; SMN2KDM4E
SCHEMBL5298071 0.72 MAOB (0.39) GPR3ALDH1A1HPGDSMN1; SMN2HSD17B10
SCHEMBL7155004 0.72 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2KDM4EGLAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317459-A1 BICYCLIC PYRROLYL AMIDES AS GLUCOGEN PHOSPHORYLASE INHIBITORS AstraZeneca AB (SE) 2003-06-11 EP disclosed
WO-2002020530-A1 BICYCLIC PYRROLYL AMIDES AS GLUCOGEN PHOSPHORYLASE INHIBITORS ASTRAZENECA AB (SE) 2002-03-14 WO disclosed