SCHEMBL7002275

SCHEMBL7002275

CCOC(=O)CCN(C)C(=O)c1cc[nH]c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.40
ALOX5 P09917 1/20 0.38
LTA4H P09960 2/20 0.38
CYP4F2 P78329 2/20 0.37
CYP4A11 Q02928 2/20 0.37
LMNA P02545 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
MAPT P10636 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
TSHR P16473 1/20 0.34
DRD2 P14416 1/20 0.34
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
TRPM8 Q7Z2W7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6997418 0.81 CDK4 (0.39) CYP4F2CYP4A11HDAC6CDK4CCND1
SCHEMBL716520 0.77 LMNA (0.53) SMN1; SMN2LTA4HCYP4F2CYP4A11LMNA
Hydrochloric Acid SCHEMBL28746969 0.76 LMNA (0.51) SMN1; SMN2LTA4HCYP4F2CYP4A11LMNA
SCHEMBL6990085 0.75 SMN1; SMN2 (0.43) SMN1; SMN2ALOX5LTA4HCYP4F2CYP4A11
SCHEMBL5162771 0.73 ALDH1A1 (0.49) SMN1; SMN2LMNAL3MBTL1MAPTTDP1
SCHEMBL3095592 0.73 LMNA (0.49) SMN1; SMN2LMNAL3MBTL1MAPTTDP1
SCHEMBL7195997 0.73 L3MBTL1 (0.43) SMN1; SMN2ALOX5LTA4HCYP4F2CYP4A11
SCHEMBL671053 0.72 CA12 (0.53) SMN1; SMN2LMNAMAPTCYP1A2CYP3A4
Hydrochloric Acid SCHEMBL27813064 0.71 CA12 (0.52) SMN1; SMN2LMNAMAPTCYP1A2CYP3A4
SCHEMBL826081 0.69 ALDH1A1 (0.45) SMN1; SMN2MAPTALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915881-B1 PYRROLOAZEPINE COMPOUNDS SUNTORY LTD (JP) 2003-01-08 EP disclosed
US-6211362-B1 CHEMICAL INTERMEDIATE FOR DRUGS SUNTORY LIMITED (JP) 2001-04-03 US disclosed
US-6187772-B1 Pyrroloazepine compounds SUNTORY LIMITED (JP) 2001-02-13 US disclosed
EP-0915881-A1 PYRROLOAZEPINE COMPOUNDS SUNTORY LIMITED (JP) 1999-05-19 EP disclosed
WO-1998041527-A1 PYRROLOAZEPINE COMPOUNDS SUNTORY LIMITED (JP) 1998-09-24 WO disclosed