SCHEMBL7003191

SCHEMBL7003191

COC(=O)c1c(O)c2cc(=O)c(OCc3ccccc3)cc-2cn1CC(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.41
LMNA P02545 1/20 0.41
NOTUM Q6P988 1/20 0.40
ERN1 O75460 1/20 0.39
PDE4A P27815 3/20 0.39
PDE4B Q07343 3/20 0.39
PDE4C Q08493 3/20 0.39
PDE4D Q08499 3/20 0.39
PDE5A O76074 2/20 0.39
SMPD1 P17405 2/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
PTGER1 P34995 1/20 0.37
PTGER4 P35408 1/20 0.37
PTGER3 P43115 1/20 0.37
PTGER2 P43116 1/20 0.37
ABCB1 P08183 1/20 0.36
PTPN1 P18031 1/20 0.36
MCL1 Q07820 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7004236 0.91 MMP2 (0.43) HPGDLMNAPTGER1ALDH1A1MAPT
SCHEMBL7556080 0.91 CRHBP (0.43) HPGDLMNANOTUMERN1PTGER1
SCHEMBL7004596 0.83 PTGER1 (0.39) PDE4APDE4BPDE4CPDE4DSMPD1
SCHEMBL7003666 0.81 PPARG (0.41) HPGDLMNAPTGER1PTGER4PTGER3
SCHEMBL7560338 0.79 CRHBP (0.43) HPGDLMNAERN1PTGER1MCL1
SCHEMBL7560366 0.77 PTGER1 (0.37) PTGER1PTGER4PTGER3PTGER2ABCB1
SCHEMBL7003154 0.68 PTPN11 (0.37) HPGDLMNAALDH1A1HTTMAPT
SCHEMBL5233228 0.68 PDE5A (0.52) HPGDLMNAPDE4APDE4BPDE4C
SCHEMBL5235849 0.68 MAPK8 (0.50) HPGDLMNAPDE4APDE4BPDE4C
SCHEMBL28448203 0.67 HPGD (0.71) HPGDLMNASMPD1HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A9 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-10-10 WO disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed