SCHEMBL7004596

SCHEMBL7004596

CC(C)Cn1cc2cc(OCc3ccccc3)c(=O)cc-2c(-c2ccccc2)c1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 7/20 0.39
PTGER4 P35408 4/20 0.39
PTGER3 P43115 4/20 0.39
PTGER2 P43116 4/20 0.39
RXRA P19793 1/20 0.37
RXRB P28702 1/20 0.37
RXRG P48443 1/20 0.37
MCL1 Q07820 2/20 0.37
ABCB1 P08183 1/20 0.37
KDM4E B2RXH2 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
SMPD1 P17405 2/20 0.36
PTPN1 P18031 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7003666 0.89 PPARG (0.41) PTGER1PTGER4PTGER3PTGER2KDM4E
SCHEMBL7560366 0.85 PTGER1 (0.37) PTGER1PTGER4PTGER3PTGER2ABCB1
SCHEMBL7003191 0.83 HPGD (0.41) PTGER1PTGER4PTGER3PTGER2MCL1
SCHEMBL7004236 0.81 MMP2 (0.43) PTGER1MRGPRX4
SCHEMBL7556080 0.80 CRHBP (0.43) PTGER1PTGER4PTGER3PTGER2MCL1
SCHEMBL7595947 0.71 DPP4 (0.39)
SCHEMBL1381646 0.70 HK2 (0.40)
SCHEMBL7560338 0.68 CRHBP (0.43) PTGER1MCL1KDM4EMRGPRX4
SCHEMBL5231509 0.67 DPP4 (0.59) PDE4APDE4BPDE4CPDE4D
SCHEMBL5234388 0.67 DPP4 (0.58)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A9 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-10-10 WO disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed