SCHEMBL7560338

SCHEMBL7560338

CCOC(=O)c1c(O)c2cc(=O)c(OCc3ccccc3)cc-2cn1CC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.43
CRHR2 Q13324 1/20 0.43
PPARG P37231 1/20 0.39
MMP2 P08253 1/20 0.39
MAPT P10636 3/20 0.38
GAA P10253 2/20 0.38
ALDH1A1 P00352 1/20 0.38
PTGER1 P34995 2/20 0.37
F2RL3 Q96RI0 1/20 0.37
LMNA P02545 2/20 0.36
HPGD P15428 1/20 0.36
PPIA P62937 2/20 0.36
MCL1 Q07820 1/20 0.36
MAOB P27338 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7004236 0.88 MMP2 (0.43) CRHBPCRHR2PPARGMMP2MAPT
SCHEMBL7007295 0.80 PTPN11 (0.37) CRHBPCRHR2MAPTGAAALDH1A1
SCHEMBL7556080 0.80 CRHBP (0.43) CRHBPCRHR2MMP2MAPTPTGER1
SCHEMBL7003191 0.79 HPGD (0.41) MAPTALDH1A1PTGER1LMNAHPGD
SCHEMBL7003666 0.78 PPARG (0.41) PPARGMMP2MAPTGAAALDH1A1
SCHEMBL7007699 0.77 CRHBP (0.39) CRHBPCRHR2MAPTGAAALDH1A1
SCHEMBL7002021 0.73 NR1H4 (0.33) PPARGALDH1A1MCL1TDP1L3MBTL1
SCHEMBL7561375 0.71 TDP1 (0.42) CRHBPCRHR2MAPTGAAALDH1A1
SCHEMBL7006171 0.68 ESR1 (0.34) GAAALDH1A1LMNAHPGDCYP2C9
SCHEMBL7004596 0.68 PTGER1 (0.39) PTGER1MCL1MRGPRX4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002062764-A9 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-10-10 WO disclosed