SCHEMBL7005503

SCHEMBL7005503

CCCCOc1c2cc(Cl)c(Cl)c(=O)c-2cn(C2CC2)c1N(C)C(=O)O

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
THRB P10828 4/20 0.32
THRA P10827 3/20 0.32
S1PR1 P21453 6/20 0.31
S1PR5 Q9H228 5/20 0.31
ESR1 P03372 1/20 0.31
S1PR3 Q99500 4/20 0.30
TAAR1 Q96RJ0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7006238 0.85 THRB (0.31) THRBTHRAS1PR1S1PR5
SCHEMBL7007555 0.82 FFAR4 (0.34) THRBTHRAESR1
SCHEMBL7006211 0.80 THRA (0.32) THRBTHRAESR1
SCHEMBL7003285 0.79 ESR1 (0.38) THRBESR1
SCHEMBL5236587 0.73 THRB (0.34) THRBTHRAS1PR1S1PR5TAAR1
SCHEMBL5234366 0.67 ALDH1A1 (0.33) THRBTHRA
SCHEMBL5234473 0.66 THRB (0.37) THRBTHRAESR1
SCHEMBL7592050 0.65 THRA (0.36) THRBTHRA
SCHEMBL5239328 0.65 CNR2 (0.36) ESR1
SCHEMBL7562047 0.65 TNF (0.37) ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed