SCHEMBL7003285

SCHEMBL7003285

CCCCOc1c2cc(Cl)c(Cl)c(=O)c-2cn(C2CC2)c1C(=O)OCC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.38
BAZ2B Q9UIF8 1/20 0.34
BAZ2A Q9UIF9 1/20 0.34
ALDH1A1 P00352 2/20 0.34
MAPK1 P28482 1/20 0.34
ADRB2 P07550 1/20 0.33
PCSK9 Q8NBP7 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
WDR5 P61964 1/20 0.32
THRB P10828 2/20 0.32
CYP1A2 P05177 2/20 0.31
NPC1 O15118 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
CYP2C19 P33261 1/20 0.31
RAB9A P51151 1/20 0.31
HTR3E A5X5Y0 1/20 0.31
GMNN O75496 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7010259 0.82 ESR1 (0.39) ESR1BAZ2BBAZ2AALDH1A1MAPK1
SCHEMBL7006414 0.81 ESR1 (0.39) ESR1BAZ2BBAZ2AALDH1A1MAPK1
SCHEMBL7006166 0.80 ESR1 (0.38) ESR1BAZ2BBAZ2AALDH1A1SMN1; SMN2
SCHEMBL7005503 0.79 THRB (0.32) ESR1THRB
SCHEMBL7006924 0.78 CRHBP (0.44) ESR1ALDH1A1SMN1; SMN2TSHR
SCHEMBL7003687 0.78 ESR1 (0.37) ESR1BAZ2BBAZ2ASMN1; SMN2THRB
SCHEMBL7000138 0.78 ESR1 (0.36) ESR1BAZ2BBAZ2A
SCHEMBL7562047 0.73 TNF (0.37) ESR1
SCHEMBL5235846 0.72 ESR1 (0.38) ESR1BAZ2BBAZ2AALDH1A1MAPK1
SCHEMBL7592050 0.68 THRA (0.36) TP53THRBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A9 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-10-10 WO disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed