SCHEMBL7006322

SCHEMBL7006322

Cc1nc(N[C@@H](C)c2ccccc2)nc(N)c1CCc1cccc(C#N)c1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 2/20 0.44
HTR7 P34969 6/20 0.43
PLK1 P53350 1/20 0.42
ADORA2B P29275 1/20 0.41
VNN1 O95497 3/20 0.38
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
DHFR P00374 1/20 0.37
GPR139 Q6DWJ6 1/20 0.37
NOS1 P29475 1/20 0.37
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
LDHA P00338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7007978 0.85 HTR7 (0.45) HTR7ADRA1DADRA1AADRA1BLDHA
SCHEMBL7014065 0.85 HTR7 (0.47) HTR7PLK1ADRA1DADRA1AADRA1B
SCHEMBL7007980 0.85 HTR7 (0.45) HTR7ADRA1DADRA1AADRA1BLDHA
SCHEMBL4383409 0.84 TLR8 (0.46) MAPK14HTR7PLK1DHFRGPR139
SCHEMBL7009364 0.81 HTR7 (0.49) HTR7ADRA1DADRA1AADRA1B
SCHEMBL7006329 0.80 F7 (0.44) HTR7LDHA
SCHEMBL4375476 0.79 HTR7 (0.65) MAPK14HTR7ADORA2BADRA1DADRA1A
SCHEMBL7007986 0.78 HTR7 (0.43) HTR7PLK1ADRA1DADRA1AADRA1B
SCHEMBL7018081 0.77 ALDH1A1 (0.46) HTR7PLK1ADRA1DADRA1AADRA1B
SCHEMBL7014716 0.77 ALDH1A1 (0.41) HTR7ADRA1DADRA1AADRA1BLDHA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1280781-A4 5-HT 7 RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2003-08-06 EP disclosed
EP-1280781-A1 5-HT 7 RECEPTOR ANTAGONISTS Bristol-Myers Squibb Company (US) 2003-02-05 EP disclosed
WO-2001085701-A1 5-HT7 RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-11-15 WO disclosed