SCHEMBL7014716

SCHEMBL7014716

COc1ccc(CCc2c(C)nc(N[C@@H](C)c3ccccc3)nc2N)cc1Br

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
MAPT P10636 1/20 0.40
KMT2A Q03164 4/20 0.39
HTR7 P34969 4/20 0.39
BCHE P06276 2/20 0.39
ACHE P22303 2/20 0.39
SOS1 Q07889 2/20 0.38
EGFR P00533 2/20 0.38
KRAS P01116 1/20 0.38
LDHA P00338 1/20 0.38
LDHB P07195 1/20 0.38
LMNA P02545 1/20 0.38
MEN1 O00255 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
ADRA1D P25100 1/20 0.37
ADRA1A P35348 1/20 0.37
ADRA1B P35368 1/20 0.37
OPRK1 P41145 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4376798 0.85 ALDH1A1 (0.43) ALDH1A1GAAPKMMAPTKMT2A
SCHEMBL7018081 0.84 ALDH1A1 (0.46) ALDH1A1KMT2AHTR7MEN1ADRA1D
SCHEMBL7007986 0.83 HTR7 (0.43) ALDH1A1HTR7SOS1EGFRKRAS
SCHEMBL7007978 0.83 HTR7 (0.45) ALDH1A1HTR7LDHAADRA1DADRA1A
SCHEMBL7007980 0.83 HTR7 (0.45) ALDH1A1HTR7LDHAADRA1DADRA1A
SCHEMBL7009364 0.81 HTR7 (0.49) HTR7ADRA1DADRA1AADRA1B
SCHEMBL7014065 0.79 HTR7 (0.47) KMT2AHTR7LDHAMEN1ADRA1D
SCHEMBL7006322 0.77 MAPK14 (0.44) HTR7LDHAADRA1DADRA1AADRA1B
SCHEMBL7006329 0.74 F7 (0.44) ALDH1A1MAPTKMT2AHTR7EGFR
SCHEMBL4381740 0.73 HTR7 (0.49) ALDH1A1GAAPKMMAPTHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1280781-A4 5-HT 7 RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2003-08-06 EP claimed
EP-1280781-A1 5-HT 7 RECEPTOR ANTAGONISTS Bristol-Myers Squibb Company (US) 2003-02-05 EP claimed
WO-2001085701-A1 5-HT7 RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-11-15 WO claimed