SCHEMBL7006705

SCHEMBL7006705

COc1cc2nc(N3CCCN(C(=O)N4CCOCC4)CC3)cc(N)c2cc1-c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.51
ALDH1A1 P00352 4/20 0.51
HSD17B10 Q99714 3/20 0.51
TP53 P04637 1/20 0.51
TSHR P16473 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
AKR1C3 P42330 2/20 0.47
HPGD P15428 2/20 0.46
LMNA P02545 1/20 0.46
HTT P42858 1/20 0.46
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7011047 0.89 KDM4E (0.47) KDM4EALDH1A1HSD17B10TP53TSHR
SCHEMBL7649027 0.88 ADRA1D (0.44) AKR1C3
SCHEMBL7013220 0.86 ADRA1A (0.56) KDM4EALDH1A1HSD17B10TP53HPGD
SCHEMBL7653453 0.85 TLR9 (0.49) KDM4EHPGD
Hydrochloric Acid SCHEMBL7652032 0.85 TLR9 (0.49) KDM4EHPGD
SCHEMBL6765566 0.83 AKR1C3 (0.45) KDM4EALDH1A1HSD17B10TP53TSHR
SCHEMBL6767075 0.83 KDM4E (0.53) KDM4EALDH1A1HSD17B10TP53TSHR
SCHEMBL7654368 0.81 EHMT2 (0.47) KDM4EALDH1A1HSD17B10TP53TSHR
SCHEMBL7014073 0.79 ADRA1A (0.56) KDM4EALDH1A1HSD17B10TP53TSHR
SCHEMBL7011919 0.79 ADRA2B (0.53) KDM4EALDH1A1HSD17B10TP53TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0875506-B1 Quinoline and quinazoline compounds useful in therapy PFIZER LTD (GB) 2003-02-26 EP disclosed