SCHEMBL7006924

SCHEMBL7006924

CCCCOc1c2cc(Cl)c(Cl)c(=O)c-2cn(Cc2ccccc2)c1C(=O)OCC

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
F2RL3 Q96RI0 1/20 0.44
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
P2RX3 P56373 4/20 0.38
TSHR P16473 1/20 0.38
P2RX7 Q99572 1/20 0.38
TDP2 O95551 1/20 0.38
NSD2 O96028 1/20 0.38
PLCG1 P19174 1/20 0.38
PAX8 Q06710 1/20 0.38
RECQL P46063 1/20 0.38
MAPK10 P53779 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
LMNA P02545 2/20 0.38
PPARG P37231 1/20 0.37
ESR1 P03372 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7006414 0.85 ESR1 (0.39) ALDH1A1KDM4ETSHRSMN1; SMN2ESR1
SCHEMBL7006166 0.84 ESR1 (0.38) CRHBPCRHR2ALDH1A1SMN1; SMN2ESR1
SCHEMBL7002598 0.84 CRHBP (0.53) CRHBPCRHR2F2RL3ALDH1A1KDM4E
SCHEMBL7003687 0.83 ESR1 (0.37) SMN1; SMN2ESR1
SCHEMBL7000138 0.82 ESR1 (0.36) ESR1
SCHEMBL7010259 0.80 ESR1 (0.39) ALDH1A1SMN1; SMN2ESR1
SCHEMBL7003285 0.78 ESR1 (0.38) ALDH1A1TSHRSMN1; SMN2ESR1
SCHEMBL7562047 0.78 TNF (0.37) P2RX3LMNAESR1
SCHEMBL7555960 0.74 TDP1 (0.38) F2RL3ALDH1A1KDM4ETSHRSMN1; SMN2
SCHEMBL5233806 0.73 MAPK8 (0.46) KDM4ETSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A9 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-10-10 WO disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed