SCHEMBL7000138

SCHEMBL7000138

CCCCCOc1c2cc(Cl)c(Cl)c(=O)c-2cn(CC(C)C)c1C(=O)OCC

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.36
BAZ2B Q9UIF8 1/20 0.34
BAZ2A Q9UIF9 1/20 0.34
AKR1C4 P17516 1/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
AKR1C1 Q04828 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GPR35 Q9HC97 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7006414 0.97 ESR1 (0.39) ESR1BAZ2BBAZ2AL3MBTL1GPR35
SCHEMBL7592050 0.89 THRA (0.36)
SCHEMBL7003687 0.88 ESR1 (0.37) ESR1BAZ2BBAZ2AL3MBTL1GPR35
SCHEMBL7006166 0.84 ESR1 (0.38) ESR1BAZ2BBAZ2AL3MBTL1
SCHEMBL7010259 0.84 ESR1 (0.39) ESR1BAZ2BBAZ2AL3MBTL1GPR35
SCHEMBL7006924 0.82 CRHBP (0.44) ESR1
SCHEMBL7004554 0.82 BAZ2B (0.39) ESR1BAZ2BBAZ2AGPR35
SCHEMBL7555501 0.79 GPR35 (0.36) BAZ2BBAZ2AGPR35
SCHEMBL7003285 0.78 ESR1 (0.38) ESR1BAZ2BBAZ2A
SCHEMBL7006211 0.77 THRA (0.32) ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A9 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-10-10 WO disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed