SCHEMBL7007036

SCHEMBL7007036

CC(C)Cn1c(=O)n(C)c(=O)c2cc(Cc3c[nH]c4ncccc34)sc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC16A1 P53985 9/20 0.57
CYP2C9 P11712 7/20 0.57
CYP3A4 P08684 7/20 0.57
GPR84 Q9NQS5 1/20 0.44
MET P08581 1/20 0.40
PDE2A O00408 4/20 0.40
PDE1A P54750 4/20 0.40
PDE1B Q01064 4/20 0.40
PDE1C Q14123 4/20 0.40
FGFR1 P11362 1/20 0.39
FGFR4 P22455 1/20 0.39
SLC16A7 O60669 1/20 0.39
MAPKAPK2 P49137 1/20 0.38
CAMK2B Q13554 1/20 0.38
HIPK4 Q8NE63 1/20 0.38
PDE5A O76074 2/20 0.38
PDE3B Q13370 2/20 0.38
PDE3A Q14432 2/20 0.38
CYP1A2 P05177 1/20 0.38
CFTR P13569 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5864831 0.82 SLC16A1 (0.58) SLC16A1CYP2C9CYP3A4PDE2APDE1A
SCHEMBL7497166 0.81 SLC16A1 (0.45) SLC16A1CYP2C9CYP3A4PDE2APDE1A
SCHEMBL7006986 0.79 SLC16A1 (0.43) SLC16A1CYP2C9CYP3A4PDE2APDE1A
SCHEMBL3833017 0.79 SLC16A1 (0.75) SLC16A1CYP2C9CYP3A4SLC16A7MAPKAPK2
SCHEMBL7008583 0.79 TBXAS1 (0.42) SLC16A1CYP2C9CYP3A4PDE2APDE1A
SCHEMBL3827986 0.78 SLC16A1 (0.73) SLC16A1CYP2C9CYP3A4SLC16A7MAPKAPK2
SCHEMBL5864692 0.77 SLC16A1 (0.56) SLC16A1CYP2C9CYP3A4SLC16A7MAPKAPK2
SCHEMBL5865214 0.77 ALDH1A1 (0.45) SLC16A1CYP2C9CYP3A4MAPKAPK2CAMK2B
SCHEMBL5864889 0.77 SLC16A1 (0.42) SLC16A1CYP2C9CYP3A4METPDE2A
SCHEMBL5864895 0.76 PDE3B (0.47) SLC16A1CYP2C9CYP3A4SLC16A7MAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1107973-B1 NOVEL THIENO[2,3-d]PYRIMIDINEDIONES, PROCESS FOR THEIR PREPARATION AND USE THEREOF IN THERAPY ASTRAZENECA AB (SE) 2003-11-05 EP claimed