SCHEMBL7007295

SCHEMBL7007295

CCOC(=O)c1c(O)c2cc(=O)c(F)cc-2cn1CC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.37
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
ALDH1A1 P00352 4/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
BCL2L1 Q07817 1/20 0.34
HPGD P15428 3/20 0.34
HSD17B10 Q99714 3/20 0.34
NPSR1 Q6W5P4 2/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
KMT2A Q03164 1/20 0.34
TSHR P16473 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7559797 0.88 ALDH1A1 (0.38) PTPN11CRHBPCRHR2ALDH1A1GAA
SCHEMBL7003154 0.86 PTPN11 (0.37) PTPN11ALDH1A1GAAMAPTBCL2L1
SCHEMBL7006666 0.84 PTPN11 (0.35) PTPN11ALDH1A1GAAMAPTBCL2L1
SCHEMBL7007699 0.83 CRHBP (0.39) PTPN11CRHBPCRHR2ALDH1A1GAA
SCHEMBL7560338 0.80 CRHBP (0.43) CRHBPCRHR2ALDH1A1GAAMAPT
SCHEMBL7556806 0.75 BAZ2B (0.38) PTPN11CRHBPCRHR2ALDH1A1GAA
SCHEMBL7006171 0.73 ESR1 (0.34) ALDH1A1GAAHPGDHSD17B10NPSR1
SCHEMBL7002285 0.73 MCL1 (0.38) PTPN11
SCHEMBL7564220 0.73 MAPT (0.38) CRHBPCRHR2ALDH1A1GAAMAPT
SCHEMBL7561375 0.73 TDP1 (0.42) CRHBPCRHR2ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A9 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-10-10 WO disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed