SCHEMBL7007318

SCHEMBL7007318

CC(C)Oc1c(F)c(F)cc(C(=O)O)c1F

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
KMT2A Q03164 1/20 0.37
KEAP1 Q14145 1/20 0.36
NFE2L2 Q16236 1/20 0.36
MAPT P10636 2/20 0.35
KDM4E B2RXH2 2/20 0.35
HTT P42858 1/20 0.35
KAT6A Q92794 2/20 0.34
RXRA P19793 1/20 0.33
RXRB P28702 1/20 0.33
DHODH Q02127 2/20 0.33
FFAR4 Q5NUL3 1/20 0.33
CES2 O00748 3/20 0.33
CES1 P23141 3/20 0.33
ASPH Q12797 1/20 0.33
KDM8 Q8N371 1/20 0.33
CXCR5 P32302 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7804048 0.84 KEAP1 (0.37) ALDH1A1KMT2AKEAP1NFE2L2MAPT
SCHEMBL8946849 0.81 KEAP1 (0.35) ALDH1A1KEAP1NFE2L2MAPTKDM4E
SCHEMBL607945 0.80 HSD17B10 (0.44) ALDH1A1KMT2AKEAP1NFE2L2MAPT
SCHEMBL2831144 0.80 HSD17B10 (0.39) KMT2AKEAP1NFE2L2MAPTKDM4E
SCHEMBL11916149 0.79 SLC6A2 (0.38) ALDH1A1MAPTKDM4EHTT
SCHEMBL9839630 0.79 KDM4E (0.46) ALDH1A1KEAP1NFE2L2MAPTKDM4E
SCHEMBL27927680 0.79 HSD17B10 (0.43) ALDH1A1KMT2AKEAP1NFE2L2MAPT
SCHEMBL9566698 0.76 KEAP1 (0.32) KEAP1NFE2L2MAPT
SCHEMBL9566679 0.76 THRA (0.46) ALDH1A1MAPTKDM4EHTT
Propylene Glycol SCHEMBL2834441 0.76 HSD17B10 (0.36) ALDH1A1KMT2AMAPTKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945435-B1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMA CO LTD (JP) 2003-08-13 EP disclosed
US-6136823-A BACTERICIDES OR VIRICIDES WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-0945435-A1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 1999-09-29 EP disclosed