SCHEMBL8613696

SCHEMBL8613696

CN1CCCC(COc2cc3c(cc2Br)CCN3)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.44
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
CDC42BPB Q9Y5S2 1/20 0.40
MAOA P21397 2/20 0.39
MAOB P27338 2/20 0.39
EGFR P00533 2/20 0.37
FGFR1 P11362 2/20 0.37
FLT1 P17948 2/20 0.37
FLT4 P35916 2/20 0.37
KDR P35968 2/20 0.37
IRAK4 Q9NWZ3 1/20 0.36
UTS2R Q9UKP6 1/20 0.35
PIK3CD O00329 1/20 0.35
PIK3R1 P27986 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
BRD4 O60885 1/20 0.35
EP300 Q09472 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8615064 0.88 ALDH1A1 (0.37) HRH3ROCK2CDC42BPBMAOAMAOB
SCHEMBL8617442 0.83 CHRNB4 (0.46)
SCHEMBL8613634 0.81 UTS2R (0.39) UTS2RALDH1A1MAPT
SCHEMBL18152767 0.78 HTR2C (0.40) HTR2AHTR2CHTR2BALDH1A1MAPT
SCHEMBL8588306 0.74 IKBKB (0.40) HRH3UTS2RHTR2AHTR2CHTR2B
SCHEMBL7096511 0.72 HRH3 (0.54) HRH3
SCHEMBL18115471 0.71 HTR2C (0.64) HTR2AHTR2CHTR2BALDH1A1MAPT
SCHEMBL8621841 0.71 HRH3 (0.44) HRH3MAOAMAOBEGFRFGFR1
SCHEMBL8656325 0.69 ALDH1A1 (0.40) HRH3ALDH1A1MAPT
SCHEMBL8792100 0.69 CHRNB4 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998050346-A2 ACETAMIDE AND UREA DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF CNS DISORDERS SMITHKLINE BEECHAM PLC (GB) 1998-11-12 WO disclosed