SCHEMBL7007897

SCHEMBL7007897

COc1ccc(C=C2C(=O)COC2=O)c(OC)c1OC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.56
SIRT1 Q96EB6 1/20 0.55
KMT2A Q03164 4/20 0.55
ALDH1A1 P00352 3/20 0.55
MAPT P10636 3/20 0.55
POLB P06746 1/20 0.55
CRHBP P24387 1/20 0.52
CRHR2 Q13324 1/20 0.52
NFE2L2 Q16236 1/20 0.50
KDM4E B2RXH2 2/20 0.49
LMNA P02545 1/20 0.49
PLA2G1B P04054 1/20 0.48
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
ATG4B Q9Y4P1 1/20 0.48
HTT P42858 3/20 0.46
MAPK1 P28482 1/20 0.46
MEN1 O00255 3/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
KDM1A O60341 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9794694 0.79 MAPK1 (0.71) MAOBKMT2AALDH1A1MAPTLMNA
SCHEMBL7008830 0.77 KDM4E (0.57) MAOBKMT2AALDH1A1MAPTCRHBP
SCHEMBL7008510 0.75 MAPT (0.71) KMT2AALDH1A1MAPTKDM4ELMNA
SCHEMBL627723 0.75 ALDH1A1 (0.63) MAOBSIRT1KMT2AALDH1A1MAPT
SCHEMBL627251 0.74 CRHBP (0.81) MAOBKMT2AALDH1A1MAPTPOLB
SCHEMBL624342 0.74 CRHBP (0.76) MAOBSIRT1KMT2AALDH1A1MAPT
SCHEMBL7004431 0.72 MAPT (0.61) MAOBKMT2AALDH1A1MAPTPOLB
SCHEMBL21599135 0.71 SIRT1 (1.00) MAOBSIRT1KMT2AALDH1A1MAPT
SCHEMBL10743231 0.70 KDM4E (0.49) KMT2AALDH1A1MAPTKDM4ERAB9A
SCHEMBL10656266 0.70 KDM4E (0.49) KMT2AALDH1A1MAPTKDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1103554-B9 Derivatives of dihydrofuro-(3,4-b)-quinolein-1-ones, process of préparation and phamaceutical compositions containing them SERVIER LAB (FR) 2003-12-17 EP disclosed
US-6548515-B1 Use as anticancer agents LES LABORATORIES SERVIER (FR) 2003-04-15 US disclosed
EP-1103554-B1 Derivatives of dihydrofuro-(3,4-b)-quinolein-1-ones, process of préparation and phamaceutical compositions containing them SERVIER LAB (FR) 2003-03-12 EP disclosed
EP-1103554-A1 Derivatives of dihydrofuro-(3,4-b)-quinolein-1-ones, process of préparation and phamaceutical compositions containing them ADIR ET COMPAGNIE (FR) 2001-05-30 EP disclosed