SCHEMBL7008752

SCHEMBL7008752

CCOC(=O)c1c(O)c2cc(Cl)c(Cl)c(=O)c-2cn1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BAZ2B Q9UIF8 1/20 0.48
BAZ2A Q9UIF9 1/20 0.48
MAPT P10636 3/20 0.42
ALDH1A1 P00352 3/20 0.42
GAA P10253 1/20 0.42
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA7 P43166 2/20 0.41
CA9 Q16790 2/20 0.41
CA14 Q9ULX7 2/20 0.41
PKM P14618 1/20 0.39
PTPN11 Q06124 2/20 0.39
ESR1 P03372 1/20 0.38
BCL2L1 Q07817 1/20 0.38
CTDSP1 Q9GZU7 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7005984 0.84 BAZ2B (0.40) BAZ2BBAZ2AMAPTALDH1A1GAA
SCHEMBL7008527 0.83 BAZ2B (0.45) BAZ2BBAZ2AMAPTALDH1A1GAA
SCHEMBL7004554 0.83 BAZ2B (0.39) BAZ2BBAZ2AMAPTALDH1A1GAA
SCHEMBL7004657 0.83 BAZ2B (0.39) BAZ2BBAZ2AMAPTALDH1A1GAA
SCHEMBL7556806 0.82 BAZ2B (0.38) BAZ2BBAZ2AMAPTALDH1A1GAA
SCHEMBL7002598 0.80 CRHBP (0.53) MAPTALDH1A1GAAPKMCYP1A2
SCHEMBL7004832 0.79 BAZ2B (0.50) BAZ2BBAZ2AMAPTALDH1A1GAA
SCHEMBL8950683 0.70 CA12 (0.60) BAZ2BBAZ2AMAPTALDH1A1CA12
SCHEMBL6834500 0.70 ALDH1A1 (0.51) BAZ2BBAZ2AMAPTALDH1A1GAA
SCHEMBL7010259 0.69 ESR1 (0.39) BAZ2BBAZ2AALDH1A1ESR1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A9 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-10-10 WO disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed