SCHEMBL7010027

SCHEMBL7010027

CCn1c(SC)nc2c(ccn2Cc2ccc(C(=O)c3ccc(C(C)(C)C)cc3O[SiH](C)C)cc2)c1=O

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 6/20 0.35
MAPT P10636 6/20 0.35
TDP1 Q9NUW8 2/20 0.34
RXFP1 Q9HBX9 5/20 0.33
THRB P10828 1/20 0.33
EPHX2 P34913 1/20 0.33
NR1H4 Q96RI1 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
ALDH1A1 P00352 2/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ENPP2 Q13822 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7017888 0.77 TP53 (0.47) TP53MAPTTDP1RXFP1THRB
Hydrochloric Acid SCHEMBL7012717 0.73 MAPT (0.39) TP53MAPTTDP1RXFP1THRB
SCHEMBL7012596 0.72 TDP1 (0.48) MAPTTDP1EPHX2NR1H4ALDH1A1
SCHEMBL7016306 0.72 TP53 (0.35) TP53MAPTTDP1RXFP1THRB
SCHEMBL7016308 0.72 CYP19A1 (0.39) TP53MAPTRXFP1TSHR
SCHEMBL7014404 0.70 TP53 (0.46) TP53MAPTTDP1RXFP1THRB
Hydrochloric Acid SCHEMBL7012711 0.69 PSMB1 (0.49) MAPTTHRBALDH1A1KDM4ETSHR
Hydrochloric Acid SCHEMBL7012709 0.69 SRC (0.37) TP53MAPTTDP1RXFP1HDAC4
SCHEMBL7019303 0.68 TP53 (0.46) TP53MAPTTDP1RXFP1THRB
SCHEMBL7015187 0.68 RAB9A (0.37) MAPTTDP1HDAC1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed