SCHEMBL7010448

SCHEMBL7010448

O=C1CCCC2=C1C(c1cccs1)c1ccccc1N2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 12/20 0.56
HSD17B10 Q99714 11/20 0.56
ALDH1A1 P00352 12/20 0.54
TSHR P16473 4/20 0.54
HPGD P15428 4/20 0.54
GAA P10253 7/20 0.54
POLB P06746 2/20 0.54
L3MBTL1 Q9Y468 2/20 0.54
ESR2 Q92731 1/20 0.54
FFAR3 O14843 1/20 0.54
ALOX15 P16050 1/20 0.52
SHMT2 P34897 1/20 0.51
USP2 O75604 3/20 0.48
HTT P42858 2/20 0.48
GLA P06280 3/20 0.48
TP53 P04637 2/20 0.48
NPSR1 Q6W5P4 2/20 0.48
MAPT P10636 2/20 0.48
LMNA P02545 1/20 0.48
CASP1 P29466 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7817207 0.85 HSD17B10 (0.65) KDM4EHSD17B10ALDH1A1TSHRHPGD
SCHEMBL7012598 0.80 GPR174 (0.59) KDM4EHSD17B10ALDH1A1GAAL3MBTL1
SCHEMBL15435872 0.77 GPR174 (0.62) KDM4EHSD17B10TSHRGAAMAPT
SCHEMBL7010637 0.76 FFAR3 (0.54) KDM4EHSD17B10ALDH1A1HPGDGAA
SCHEMBL2998592 0.71 KDM4E (1.00) KDM4EHSD17B10ALDH1A1TSHRHPGD
SCHEMBL3326098 0.69 KDM4E (0.80) KDM4EHSD17B10ALDH1A1TSHRHPGD
SCHEMBL3242208 0.69 FFAR3 (0.70) KDM4EHSD17B10ALDH1A1TSHRHPGD
SCHEMBL3324020 0.69 KDM4E (0.78) KDM4EHSD17B10ALDH1A1TSHRHPGD
SCHEMBL16583705 0.69 HSD17B10 (0.67) KDM4EHSD17B10ALDH1A1TSHRHPGD
SCHEMBL17792787 0.68 SHMT2 (1.00) KDM4EHSD17B10ALDH1A1TSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1103554-B9 Derivatives of dihydrofuro-(3,4-b)-quinolein-1-ones, process of préparation and phamaceutical compositions containing them SERVIER LAB (FR) 2003-12-17 EP claimed
EP-1103554-B1 Derivatives of dihydrofuro-(3,4-b)-quinolein-1-ones, process of préparation and phamaceutical compositions containing them SERVIER LAB (FR) 2003-03-12 EP claimed
EP-1103554-B9 Derivatives of dihydrofuro-(3,4-b)-quinolein-1-ones, process of préparation and phamaceutical compositions containing them SERVIER LAB (FR) 2003-12-17 EP disclosed
EP-1103554-B1 Derivatives of dihydrofuro-(3,4-b)-quinolein-1-ones, process of préparation and phamaceutical compositions containing them SERVIER LAB (FR) 2003-03-12 EP disclosed