SCHEMBL7014308

SCHEMBL7014308

O=C(c1ccc(Cl)cc1)c1ccc(CSc2nc3ccccc3c(=O)n2CF)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.59
TBXA2R P21731 5/20 0.59
CYP1A2 P05177 3/20 0.58
CYP2C9 P11712 3/20 0.58
CYP2C19 P33261 3/20 0.58
CYP2D6 P10635 2/20 0.58
MAPT P10636 1/20 0.58
NPSR1 Q6W5P4 1/20 0.58
CA12 O43570 2/20 0.57
CA1 P00915 2/20 0.57
CA2 P00918 2/20 0.57
CA9 Q16790 2/20 0.57
MEN1 O00255 4/20 0.56
KMT2A Q03164 4/20 0.56
PTGDR2 Q9Y5Y4 1/20 0.56
HDAC3 O15379 1/20 0.53
HDAC4 P56524 1/20 0.53
HDAC1 Q13547 1/20 0.53
HDAC7 Q8WUI4 1/20 0.53
HDAC2 Q92769 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7015339 0.85 KMT2A (0.68) DRD2TBXA2RCYP1A2CYP2C9CYP2C19
SCHEMBL7018117 0.77 TDP1 (0.64) DRD2TBXA2RCYP1A2CYP2C9CYP2C19
SCHEMBL7013706 0.77 KMT2A (0.68) MAPTCA12CA1CA2CA9
SCHEMBL7015464 0.75 KMT2A (0.60) DRD2TBXA2RCYP1A2CYP2C9CYP2C19
SCHEMBL7014540 0.75 DRD2 (0.52) DRD2TBXA2RCYP1A2CYP2C9CYP2C19
SCHEMBL7013210 0.74 MEN1 (0.53) DRD2TBXA2RCYP1A2CYP2C9CYP2C19
SCHEMBL7012108 0.74 MAOB (0.84) MAPTMEN1KMT2AALDH1A1
SCHEMBL8646764 0.73 L3MBTL1 (0.68) CYP1A2CYP2C9CYP2C19CYP2D6MAPT
SCHEMBL7018370 0.72 MEN1 (0.50) DRD2TBXA2RCYP1A2CYP2C9CYP2C19
SCHEMBL7019775 0.72 MEN1 (0.58) CYP1A2CYP2C9CYP2C19CYP2D6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed