SCHEMBL7010850

SCHEMBL7010850

COC(=O)c1cccc2nc(SCc3ccc(C(=O)c4ccc(Cl)cc4)cc3)n(C)c(=O)c12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.55
TBXA2R P21731 6/20 0.55
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
RAB9A P51151 1/20 0.50
MAPT P10636 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
PTGDR2 Q9Y5Y4 2/20 0.45
THRB P10828 2/20 0.45
TP53 P04637 2/20 0.45
HDAC3 O15379 2/20 0.44
HDAC4 P56524 2/20 0.44
HDAC1 Q13547 2/20 0.44
HDAC7 Q8WUI4 2/20 0.44
HDAC2 Q92769 2/20 0.44
HDAC10 Q969S8 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7018370 0.85 MEN1 (0.50) DRD2TBXA2RMEN1KMT2AMAPT
SCHEMBL7014355 0.85 DRD2 (0.50) DRD2TBXA2RMEN1KMT2ARAB9A
SCHEMBL7014213 0.85 DRD2 (0.48) DRD2TBXA2RMEN1KMT2AMAPT
SCHEMBL7013547 0.84 PTGDR2 (0.52) DRD2TBXA2RMEN1KMT2ARAB9A
SCHEMBL7015339 0.80 KMT2A (0.68) DRD2TBXA2RMEN1KMT2AMAPT
SCHEMBL7011506 0.80 MEN1 (0.55) MEN1KMT2AMAPTCYP1A2CYP2D6
SCHEMBL7014904 0.79 LMNA (0.45) DRD2TBXA2RMEN1KMT2ARAB9A
SCHEMBL7018222 0.79 TDP1 (0.49) DRD2TBXA2RMEN1KMT2AMAPT
SCHEMBL7014463 0.79 MEN1 (0.49) DRD2TBXA2RMEN1KMT2ARAB9A
SCHEMBL7015237 0.78 MEN1 (0.45) DRD2TBXA2RMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed