SCHEMBL7019103

SCHEMBL7019103

CSc1nc2[nH]ccc2c(=O)n1CCOC(C)=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
ADORA2B P29275 2/20 0.40
MAPT P10636 2/20 0.38
LMNA P02545 2/20 0.37
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
IDO1 P14902 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
GAA P10253 3/20 0.36
NEK1 Q96PY6 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
POLB P06746 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7010831 0.81 ALDH1A1 (0.42) ALDH1A1ADORA2BSMN1; SMN2NPSR1
SCHEMBL7018141 0.79 MAPK1 (0.40) ALDH1A1MAPTLMNAKDM4EMEN1
SCHEMBL13257531 0.70 LMNA (0.44) ALDH1A1LMNAKDM4ESMN1; SMN2POLB
SCHEMBL7015802 0.69 NEK1 (0.39) ALDH1A1HTTNEK1JAK2JAK1
SCHEMBL7008875 0.68 TP53 (0.42) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL13863953 0.67 ALDH1A1 (0.73) ALDH1A1ADORA2BMAPTKDM4ETDP1
SCHEMBL2564399 0.65 FADS1 (0.48) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL2570522 0.64 POLB (0.48) ALDH1A1LMNAMEN1KMT2APOLB
SCHEMBL3829770 0.64 TSHR (0.64) ALDH1A1KDM4EMEN1KMT2AGAA
SCHEMBL13266383 0.64 TP53 (0.35) LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed