SCHEMBL7016241

SCHEMBL7016241

CC(=O)OCCn1cnc2c(c(C)cn2Cc2ccc(C(=O)c3ccc(Cl)cc3)cc2)c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.43
ADORA2B P29275 2/20 0.43
TP53 P04637 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MAPK1 P28482 3/20 0.41
LMNA P02545 1/20 0.41
ALDH1A1 P00352 4/20 0.40
HSD17B10 Q99714 3/20 0.40
KDM4E B2RXH2 2/20 0.40
KMT2A Q03164 3/20 0.39
TSHR P16473 3/20 0.39
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39
MEN1 O00255 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
RECQL P46063 1/20 0.37
MAPK10 P53779 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7020188 0.88 LMNA (0.46) SMN1; SMN2TP53TDP1MAPK1LMNA
SCHEMBL7017298 0.85 TP53 (0.46) SMN1; SMN2TP53TDP1MAPK1LMNA
SCHEMBL7015987 0.84 TP53 (0.47) SMN1; SMN2TP53TDP1MAPK1LMNA
SCHEMBL7016238 0.80 MAPT (0.43) SMN1; SMN2TP53TDP1MAPK1LMNA
SCHEMBL7020184 0.79 TP53 (0.44) SMN1; SMN2TP53TDP1MAPK1LMNA
SCHEMBL7021271 0.77 CYP19A1 (0.41) SMN1; SMN2TP53TDP1MAPK1LMNA
SCHEMBL7016056 0.76 THRB (0.47) SMN1; SMN2TP53ALDH1A1KMT2ATSHR
SCHEMBL7008880 0.76 TP53 (0.37) SMN1; SMN2TP53TDP1MAPK1LMNA
SCHEMBL7017354 0.75 THRB (0.48) SMN1; SMN2TP53KMT2ATSHRMEN1
SCHEMBL7019393 0.75 HTT (0.42) SMN1; SMN2TP53ALDH1A1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed