SCHEMBL7019393

SCHEMBL7019393

CCn1cnc2c(c(C)cn2Cc2ccc(C(=O)c3ccc(C(F)(F)F)cc3)cc2)c1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.42
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MMP13 P45452 1/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
NR3C1 P04150 1/20 0.40
SRD5A2 P31213 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KMT2A Q03164 1/20 0.39
ABCC8 Q09428 1/20 0.38
KCNJ11 Q14654 1/20 0.38
MAPT P10636 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7016056 0.90 THRB (0.47) HTTALDH1A1SMN1; SMN2KMT2AMAPT
SCHEMBL7017298 0.89 TP53 (0.46) ALDH1A1CYP1A2CYP3A4CYP2C19SMN1; SMN2
SCHEMBL7021271 0.89 CYP19A1 (0.41) HTTKDM4ESMN1; SMN2KMT2AMAPT
SCHEMBL7008880 0.85 TP53 (0.37) ALDH1A1CYP1A2CYP3A4CYP2C19SMN1; SMN2
SCHEMBL7020188 0.79 LMNA (0.46) KDM4EALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL7017354 0.78 THRB (0.48) HTTSMN1; SMN2KMT2AMAPTPOLB
SCHEMBL7015987 0.77 TP53 (0.47) KDM4EALDH1A1CYP1A2CYP3A4CYP2C19
Hydrochloric Acid SCHEMBL7015357 0.76 ALDH1A1 (0.36) HTTKDM4EALDH1A1MMP13CYP3A4
Hydrochloric Acid SCHEMBL7015359 0.76 SMN1; SMN2 (0.48) KDM4EALDH1A1SMN1; SMN2KMT2AMAPT
SCHEMBL7014131 0.75 ABCC8 (0.70) HTTALDH1A1SMN1; SMN2ABCC8KCNJ11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed